SCHEMBL10370353

SCHEMBL10370353

CC(=O)CCCC(C#N)(Cc1cccnc1)c1ccc(Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.40
FNTA P49354 1/20 0.39
FNTB P49356 1/20 0.39
CYP19A1 P11511 3/20 0.39
FDPS P14324 4/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HIF1A Q16665 1/20 0.37
GPR119 Q8TDV5 1/20 0.37
HTT P42858 2/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
TBXAS1 P24557 1/20 0.36
BTN3A1 O00481 1/20 0.36
PDE3A Q14432 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10372451 0.85 TDP1 (0.45) CYP19A1FDPSCYP1A2CYP3A4CYP2C9
SCHEMBL10372391 0.83 CYP19A1 (0.42) CYP19A1FDPSCYP1A2CYP3A4CYP2C9
SCHEMBL10370926 0.83 CYP19A1 (0.41) KMT2ACYP19A1FDPSCYP1A2CYP3A4
SCHEMBL10370398 0.82 NR1H3 (0.41) KMT2ACYP19A1FDPSCYP1A2CYP3A4
SCHEMBL10369963 0.81 CYP19A1 (0.41) CYP19A1FDPSCYP1A2CYP3A4CYP2C9
SCHEMBL10370475 0.81 CYP19A1 (0.44) CYP19A1FDPSCYP1A2CYP3A4CYP2C9
SCHEMBL10372324 0.81 CYP19A1 (0.43) CYP19A1HTTALDH1A1SMN1; SMN2
SCHEMBL10369609 0.81 CYP3A4 (0.44) CYP19A1FDPSCYP1A2CYP3A4CYP2C9
SCHEMBL10371540 0.78 NPC1 (0.41) KMT2ACYP19A1CYP1A2CYP3A4CYP2C9
SCHEMBL10371112 0.77 CYP3A4 (0.46) CYP19A1CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0214793-B1 (2-CYANO-2-ARYLETHYL)PYRIDINES, THEIR PREPARATION AND USE AS FUNGICIDES ROHM AND HAAS COMPANY (US) 1990-06-13 EP disclosed
US-4933339-A PHYTOPATHOGENS ROHM AND HAAS COMPANY (US) 1990-06-12 US disclosed
EP-0214793-A1 (2-Cyano-2-arylethyl)pyridines, their preparation and use as fungicides ROHM AND HAAS COMPANY (US) 1987-03-18 EP disclosed