SCHEMBL10370398

SCHEMBL10370398

N#CC(CCc1ccc(Cl)cc1)(Cc1cccnc1)c1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 2/20 0.41
NR1D1 P20393 1/20 0.41
CYP19A1 P11511 6/20 0.40
CYP3A4 P08684 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HIF1A Q16665 1/20 0.39
MAPT P10636 1/20 0.38
FDPS P14324 2/20 0.37
CYP3A5 P20815 2/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10369609 0.96 CYP3A4 (0.44) NR1H3NR1D1CYP19A1CYP3A4CYP1A2
SCHEMBL10371112 0.95 CYP3A4 (0.46) NR1H3NR1D1CYP19A1CYP3A4CYP1A2
SCHEMBL10371061 0.91 NR1D1 (0.40) NR1D1CYP19A1CYP3A4CYP3A5KMT2A
SCHEMBL10371540 0.91 NPC1 (0.41) NR1H3NR1D1CYP19A1CYP3A4CYP1A2
SCHEMBL10372324 0.87 CYP19A1 (0.43) NR1H3NR1D1CYP19A1
SCHEMBL9804822 0.86 CYP19A1 (0.42) CYP19A1CYP3A4CYP3A5
SCHEMBL10370475 0.84 CYP19A1 (0.44) NR1H3NR1D1CYP19A1CYP3A4CYP1A2
SCHEMBL10369963 0.84 CYP19A1 (0.41) NR1H3NR1D1CYP19A1CYP3A4CYP1A2
SCHEMBL10372451 0.84 TDP1 (0.45) NR1H3NR1D1CYP19A1CYP3A4CYP1A2
SCHEMBL10405109 0.84 CYP3A4 (0.40) CYP19A1CYP3A4CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0214793-B1 (2-CYANO-2-ARYLETHYL)PYRIDINES, THEIR PREPARATION AND USE AS FUNGICIDES ROHM AND HAAS COMPANY (US) 1990-06-13 EP disclosed
US-4933339-A PHYTOPATHOGENS ROHM AND HAAS COMPANY (US) 1990-06-12 US disclosed
EP-0214793-A1 (2-Cyano-2-arylethyl)pyridines, their preparation and use as fungicides ROHM AND HAAS COMPANY (US) 1987-03-18 EP disclosed