SCHEMBL10370593

SCHEMBL10370593

CN(C)c1ccc2sc(S(N)(=O)=O)cc2c1

nearest known ligand 0.62

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
CA2 P00918 20/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2088019 0.78 CA2 (0.65) CA2
SCHEMBL10370434 0.77 CA2 (1.00) CA2
SCHEMBL10368067 0.76 CA2 (0.56) CA2
SCHEMBL10369727 0.75 CA2 (0.75) CA2
SCHEMBL2088451 0.75 CA2 (0.65) CA2
SCHEMBL10368289 0.75 CA2 (1.00) CA2
SCHEMBL2087596 0.74 CA2 (1.00) CA2
SCHEMBL10369174 0.73 CA2 (1.00) CA2
SCHEMBL10371815 0.72 CA2 (0.63) CA2
SCHEMBL792780 0.72 CA2 (1.00) CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129478-B1 2-SULFAMOYLBENZO (B) THIOPHENE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITION FOR THE TREATMENT OF ELEVATED INTRAOCULAR PRESSURE MERCK & CO. INC. (US) 1990-01-17 EP disclosed
US-4788192-A TOPICALLY APPLYING; FOR GLAUCOMA MERCK & CO., INC. (US) 1988-11-29 US disclosed
US-4668697-A Elevated intraocular pressure lowering benzo-[b]-thiophene-2-sulfonamide derivatives, compositions, and method of use therefor MERCK & CO., INC. (US) 1987-05-26 US disclosed
EP-0129478-A2 2-Sulfamoylbenzo (b) thiophene derivatives, their preparation and pharmaceutical composition for the treatment of elevated intraocular pressure MERCK & CO. INC. (US) 1984-12-27 EP disclosed