SCHEMBL10371018

SCHEMBL10371018

c1ccc2c(c1)O[C@@H]1CNC[C@H]1O2

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 3/20 0.39
CHRNA3 P32297 3/20 0.39
NISCH Q9Y2I1 1/20 0.38
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.36
ITGB2 P05107 1/20 0.36
ICAM1 P05362 1/20 0.36
ITGAL P20701 1/20 0.36
OXTR P30559 1/20 0.35
HTR6 P50406 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10371015 1.00 CHRNB4 (0.39) CHRNB4CHRNA3NISCHCHRNB2CHRNA4
SCHEMBL10371016 1.00 CHRNB4 (0.39) CHRNB4CHRNA3NISCHCHRNB2CHRNA4
Hydrochloric Acid SCHEMBL10977838 0.98 CHRNB4 (0.38) CHRNB4CHRNA3NISCHCHRNB2CHRNA4
SCHEMBL11959914 0.85 HTR6 (0.43) NISCHHTR6
SCHEMBL18204707 0.79 HTR6 (0.42) CHRNB4CHRNA3HTR6
Hydrochloric Acid SCHEMBL18204598 0.78 HTR6 (0.44) CHRNB4CHRNA3HTR6
SCHEMBL10375109 0.76 AHR (0.40) HTR6
SCHEMBL10375117 0.76 BRD4 (0.36) CHRNB4CHRNA3CHRNB2CHRNA4HTR6
SCHEMBL10509903 0.76 CHRM2 (0.45) NISCHCHRNB2CHRNA4OXTR
Fluparoxan SCHEMBL7173629 0.76 SLC6A2 (0.38) CHRNB2CHRNA4HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4496579-A AMINATION WITH AMMONIA OR PRIMARY AMINE; ANTIDEPRESANT GLAXO GROUP LIMITED (GB) 1985-01-29 US claimed
EP-0221725-B1 PROCESS FOR PREPARING HETEROCYCLIC COMPOUNDS GLAXO GROUP LIMITED (GB) 1990-08-08 EP disclosed
US-4496579-A AMINATION WITH AMMONIA OR PRIMARY AMINE; ANTIDEPRESANT GLAXO GROUP LIMITED (GB) 1985-01-29 US disclosed