SCHEMBL10372123

SCHEMBL10372123

COc1cnc(CSc2nc3cc(OC(F)(F)F)ccc3[nH]2)c(C)c1OCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 1/20 0.49
CYP2D6 P10635 8/20 0.47
CYP2C9 P11712 8/20 0.47
CYP2C19 P33261 8/20 0.47
CYP3A4 P08684 7/20 0.47
CYP2E1 P05181 7/20 0.47
CYP2C8 P10632 7/20 0.47
CYP2B6 P20813 7/20 0.47
CYP1A2 P05177 6/20 0.44
RAB9A P51151 5/20 0.44
NPC1 O15118 4/20 0.44
SMN1; SMN2 Q16637 3/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
ATP1A1 P05023 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10370822 0.94 BRS3 (0.51) BRS3CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL10372557 0.93 ATP4A (0.49) BRS3CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL10371409 0.91 CYP2D6 (0.51) BRS3CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL10371942 0.90 BRS3 (0.49) BRS3CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL6457331 0.90 BRS3 (0.57) BRS3CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL10373587 0.88 BRS3 (0.50) BRS3CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL10370611 0.87 ATP4A (0.49) BRS3CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL10371882 0.87 CYP2D6 (0.49) BRS3CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL10370946 0.86 CYP2E1 (0.49) CYP2D6CYP2C9CYP2C19CYP3A4CYP2E1
SCHEMBL10371431 0.85 CYP2D6 (0.52) BRS3CYP2D6CYP2C9CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0390842-A1 NOVEL BENZIMIDAZOLE DERIVATIVES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1990-10-10 EP disclosed
WO-1989005299-A1 NOVEL BENZIMIDAZOLE DERIVATIVES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1989-06-15 WO disclosed