SCHEMBL10372124

SCHEMBL10372124

COc1c(OCc2ccccc2)cnc(CSc2nc3cc(OC(F)F)ccc3[nH]2)c1C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 1/20 0.51
CYP2D6 P10635 9/20 0.48
CYP2C9 P11712 9/20 0.48
CYP2C19 P33261 9/20 0.48
CYP2E1 P05181 8/20 0.48
CYP2C8 P10632 8/20 0.48
CYP2B6 P20813 8/20 0.48
CYP3A4 P08684 8/20 0.48
ATP1A1 P05023 3/20 0.47
ATP1B1 P05026 3/20 0.47
ATP1A3 P13637 3/20 0.47
ATP1B2 P14415 3/20 0.47
ATP4A P20648 3/20 0.47
ATP1A2 P50993 3/20 0.47
ATP4B P51164 3/20 0.47
ATP1B3 P54709 3/20 0.47
FXYD2 P54710 3/20 0.47
ATP1A4 Q13733 3/20 0.47
CYP1A2 P05177 7/20 0.46
NPC1 O15118 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10371942 0.94 BRS3 (0.49) BRS3CYP2D6CYP2C9CYP2C19CYP2E1
SCHEMBL10370611 0.91 ATP4A (0.49) BRS3CYP2D6CYP2C9CYP2C19CYP2E1
SCHEMBL6882439 0.90 BRS3 (0.57) BRS3CYP2D6CYP2C9CYP2C19CYP2E1
SCHEMBL10370822 0.90 BRS3 (0.51) BRS3CYP2D6CYP2C9CYP2C19CYP2E1
SCHEMBL10370950 0.90 BRS3 (0.51) BRS3CYP2D6CYP2C9CYP2C19CYP2E1
SCHEMBL10373587 0.89 BRS3 (0.50) BRS3CYP2D6CYP2C9CYP2C19CYP2E1
SCHEMBL10373409 0.88 BRS3 (0.49) BRS3CYP2D6CYP2C9CYP2C19CYP2E1
SCHEMBL10371414 0.88 BRS3 (0.49) BRS3CYP2D6CYP2C9CYP2C19CYP2E1
SCHEMBL10371431 0.88 CYP2D6 (0.52) BRS3CYP2D6CYP2C9CYP2C19CYP2E1
SCHEMBL10370886 0.87 CYP2C9 (0.49) BRS3CYP2D6CYP2C9CYP2C19CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0390842-A1 NOVEL BENZIMIDAZOLE DERIVATIVES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1990-10-10 EP disclosed
WO-1989005299-A1 NOVEL BENZIMIDAZOLE DERIVATIVES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1989-06-15 WO disclosed