SCHEMBL10372129

SCHEMBL10372129

COSc1ccc(C(=O)O)c(O)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.50
CA12 O43570 3/20 0.50
CA1 P00915 3/20 0.50
CA2 P00918 3/20 0.50
CA7 P43166 3/20 0.50
CA9 Q16790 3/20 0.50
CA14 Q9ULX7 3/20 0.50
TSHR P16473 1/20 0.50
MCL1 Q07820 1/20 0.47
KDM4E B2RXH2 5/20 0.47
MAPT P10636 2/20 0.47
PTPN1 P18031 2/20 0.47
CYP3A4 P08684 2/20 0.47
GAA P10253 1/20 0.47
ESR2 Q92731 1/20 0.47
HNF4A P41235 1/20 0.44
ACMSD Q8TDX5 1/20 0.44
MYC P01106 2/20 0.44
KLKB1 P03952 1/20 0.44
CTSB P07858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11201624 0.98 ALDH1A1 (0.48) ALDH1A1CA12CA1CA2CA7
SCHEMBL3175665 0.86 MCL1 (0.66) ALDH1A1CA12CA1CA2CA7
SCHEMBL10374434 0.84 CA12 (0.61) ALDH1A1CA12CA1CA2CA7
SCHEMBL10373933 0.81 ALDH1A1 (0.57) ALDH1A1TSHRKDM4EMAPTGAA
SCHEMBL2956403 0.79 ALDH1A1 (0.55) ALDH1A1CA12CA1CA2CA7
SCHEMBL3161431 0.79 MCL1 (0.72) ALDH1A1CA12CA1CA2CA7
SCHEMBL15220064 0.79 ALDH1A1 (0.59) ALDH1A1CA12CA1CA2CA7
SCHEMBL10372975 0.77 LCK (0.51) ALDH1A1CA12CA1CA2CA7
SCHEMBL9117526 0.76 ALDH1A1 (0.52) ALDH1A1CA12CA1CA2CA7
SCHEMBL10398143 0.76 ALDH1A1 (0.57) ALDH1A1CA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0187487-B1 BENZOTHIOPHENES AND BENZOFURANS HAVING ANTIALLERGIC ACTIVITY WARNER-LAMBERT COMPANY (US) 1990-08-29 EP disclosed
US-4703053-A Benzothiophenes and benzofurans and antiallergic use thereof WARNER-LAMBERT COMPANY (US) 1987-10-27 US disclosed
EP-0187487-A1 Benzothiophenes and benzofurans having antiallergic activity WARNER-LAMBERT COMPANY (US) 1986-07-16 EP disclosed
US-4539412-A ANTITUMOR AGENTS RENSSELAER POLYTECHNIC INSTITUTE (US) 1985-09-03 US disclosed