SCHEMBL10375434

SCHEMBL10375434

COC(=O)c1c(C)nc(-c2ccccc2)nc1-c1cc([N+](=O)[O-])ccc1N1CCN(C)CC1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.50
WDR5 P61964 9/20 0.50
GAA P10253 3/20 0.50
LMNA P02545 2/20 0.50
POLB P06746 2/20 0.48
KMT2A Q03164 1/20 0.48
HTT P42858 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MAPK1 P28482 1/20 0.44
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10867553 0.91 ALDH1A1 (0.53) ALDH1A1WDR5GAALMNAPOLB
SCHEMBL10867548 0.91 ALDH1A1 (0.53) ALDH1A1WDR5GAALMNAPOLB
SCHEMBL10375265 0.83 KMT2A (0.46) ALDH1A1GAALMNAKMT2AHTT
SCHEMBL10375348 0.82 KMT2A (0.43) ALDH1A1LMNAKMT2AMAPK1CYP2D6
SCHEMBL10375262 0.80 KMT2A (0.41) ALDH1A1KMT2A
SCHEMBL10375282 0.78 ALDH1A1 (0.55) ALDH1A1GAAPOLBKMT2A
SCHEMBL282589 0.76 ALDH1A1 (0.62) ALDH1A1WDR5GAALMNAPOLB
SCHEMBL10375516 0.74 KDM4E (0.54) ALDH1A1GAALMNAKMT2AHTT
SCHEMBL10375206 0.73 PDE4D (0.56) ALDH1A1LMNAPOLBMAPK1
SCHEMBL10375294 0.73 KMT2A (0.48) ALDH1A1GAALMNAKMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0169712-B1 NEW PYRIMIDINE DERIVATIVES, PROCESSES FOR PREPARATION THEREOF AND COMPOSITION CONTAINING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-12-12 EP disclosed
US-4698340-A TREATMENT OF CEREBROVASCULAR DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1987-10-06 US disclosed
EP-0169712-A2 New pyrimidine derivatives, processes for preparation thereof and composition containing the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1986-01-29 EP disclosed