SCHEMBL1037803

SCHEMBL1037803

COCCCCOc1ccc([C@H]2[C@H](O[Si](C(C)C)(C(C)C)C(C)C)CN(C(=O)O)C(Cc3ccccc3)[C@@H]2OCc2ccc3c(c2)N(CCCOC)C(=O)CO3)cc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
REN P00797 5/20 0.38
CYP3A4 P08684 5/20 0.37
TSHR P16473 2/20 0.34
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
MAPT P10636 3/20 0.33
CHRM1 P11229 1/20 0.32
SMPD1 P17405 1/20 0.32
HTR1A P08908 4/20 0.32
HTR1D P28221 4/20 0.32
HTR1B P28222 4/20 0.32
CYP1A2 P05177 3/20 0.32
CYP2C9 P11712 3/20 0.32
CYP2C19 P33261 3/20 0.32
CYP2D6 P10635 2/20 0.32
POLB P06746 2/20 0.31
HSD17B10 Q99714 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3274719 0.94 REN (0.36) RENCYP3A4TSHRMAPTCHRM1
SCHEMBL1037840 0.89 REN (0.33) RENPPARGPPARA
SCHEMBL3949181 0.85 REN (0.39) RENCYP3A4TSHRPPARGPPARA
SCHEMBL3906325 0.84 REN (0.40) RENCYP3A4TSHRPPARGPPARA
SCHEMBL1037801 0.84 REN (0.39) RENCYP3A4TSHRPPARGPPARA
SCHEMBL1037108 0.83 REN (0.35) REN
SCHEMBL1034992 0.81 MAPT (0.39) RENCYP3A4TSHRMAPTCHRM1
SCHEMBL3911082 0.81 MAPT (0.40) RENCYP3A4TSHRMAPTCHRM1
SCHEMBL1036573 0.81 MAPT (0.41) RENCYP3A4TSHRMAPTCHRM1
SCHEMBL2682976 0.80 REN (0.36) RENCYP3A4TSHRMAPTHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049514-B1 NITRATE ESTERS OF PIPERIDINES NOVARTIS AG (CH) 2011-01-26 EP disclosed