SCHEMBL10378409

SCHEMBL10378409

CCOC(=O)CC[C@H](NC(=O)c1ccc(NCc2c(C)nc3nc(N)nc(N)c3c2C)cc1)C(=O)OCC

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DHFR P00374 7/20 0.50
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TYMS P04818 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10379292 0.93 DHFR (0.49) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL10379119 0.92 DHFR (0.49) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL10378274 0.90 DHFR (0.48) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL10379170 0.86 DHFR (0.45) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL10379275 0.86 DHFR (0.45) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL12692389 0.86 DHFR (0.55) DHFR
SCHEMBL10378171 0.86 DHFR (0.44) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL10378082 0.85 DHFR (0.59) DHFRTYMS
SCHEMBL10378079 0.85 DHFR (0.59) DHFRTYMS
SCHEMBL14027296 0.82 DHFR (0.55) DHFRKDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0377031-A1 5-DEAZA-5,7-DISUBSTITUTED-AMINOPTERIN ANALOGUES Sloan-Kettering Institute For Cancer Research (US) 1990-07-11 EP claimed
WO-1990000172-A1 5-DEAZA-5,7-DISUBSTITUTED-AMINOPTERIN ANALOGUES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-01-11 WO claimed