SCHEMBL1037994

SCHEMBL1037994

Cc1noc(NC(=O)N2CCC(=Cc3cccc(OC4CCC(F)(F)CC4)c3)CC2)c1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.42
CYP2D6 P10635 5/20 0.42
FAAH O00519 3/20 0.39
GABRA1 P14867 1/20 0.39
ADRA2C P18825 1/20 0.39
CNR1 P21554 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
CNR2 P34972 1/20 0.39
HTR2B P41595 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
OGA O60502 1/20 0.36
EPHX2 P34913 1/20 0.34
ALDH1A1 P00352 1/20 0.33
GPR119 Q8TDV5 2/20 0.33
POLB P06746 1/20 0.33
PKM P14618 1/20 0.33
NAMPT P43490 1/20 0.33
SLC5A7 Q9GZV3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1036941 0.93 CYP3A4 (0.40) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL1037033 0.88 CYP3A4 (0.42) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL1075874 0.84 CYP3A4 (0.43) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL1037321 0.82 POLB (0.33) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL1037320 0.82 POLB (0.33) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL6522790 0.81 PDE2A (0.33) FAAHOGAPOLB
SCHEMBL1011604 0.81 CYP3A4 (0.49) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL1075244 0.81 CYP3A4 (0.45) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL1036429 0.81 CYP3A4 (0.42) CYP3A4CYP2D6FAAHGABRA1ADRA2C
SCHEMBL1036041 0.81 CYP3A4 (0.44) CYP3A4CYP2D6FAAHGABRA1ADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2276738-A1 ETHER BENZYLIDENE PIPERIDINE 5-MEMBERED ARYL CARBOXAMIDE COMPOUNDS USEFUL AS FAAH INHIBITORS Pfizer Inc. (US) 2011-01-26 EP disclosed
WO-2009127943-A1 ETHER BENZYLIDENE PIPERIDINE 5-MEMBERED ARYL CARBOXAMIDE COMPOUNDS USEFUL AS FAAH INHIBITORS PFIZER INC. (US) 2009-10-22 WO disclosed