SCHEMBL10399151

SCHEMBL10399151

C=C/C=C(/C(N)=O)c1ccc(OC)cc1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.55
CA2 P00918 6/20 0.55
PARP10 Q53GL7 2/20 0.55
PARP1 P09874 1/20 0.55
PARP2 Q9UGN5 1/20 0.55
PARP4 Q9UKK3 1/20 0.55
MAPK1 P28482 1/20 0.50
RAB9A P51151 1/20 0.50
HSD17B10 Q99714 1/20 0.50
CES2 O00748 2/20 0.48
CES1 P23141 2/20 0.48
PKM P14618 1/20 0.46
MAPT P10636 1/20 0.46
PRSS1 P07477 1/20 0.46
PRSS2 P07478 1/20 0.46
PRSS3 P35030 1/20 0.46
PLK1 P53350 1/20 0.43
TGM2 P21980 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10399155 1.00 CA1 (0.55) CA1CA2PARP10PARP1PARP2
SCHEMBL2813142 0.85 CA1 (0.53) CA1CA2PARP10PARP1PARP2
SCHEMBL2813135 0.85 CA1 (0.53) CA1CA2PARP10PARP1PARP2
SCHEMBL27766998 0.80 EPHX2 (0.41) RAB9A
SCHEMBL14678383 0.79 CA1 (0.58) CA1CA2PARP10PARP1PARP2
SCHEMBL27909884 0.77 AKT1 (0.47) CA1CA2PARP1MAPK1HSD17B10
SCHEMBL27766838 0.75 HDAC3 (0.44) PRSS1PRSS2PRSS3
SCHEMBL10685379 0.74 ALDH1A1 (0.57) CA1CA2PARP10PARP1PARP2
SCHEMBL24205454 0.74 CA1 (0.51) CA1CA2PARP10PARP1PARP2
SCHEMBL30924784 0.74 MAPT (0.47) CA1CA2PARP10PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4975438-A ANTICOAGULANT HOFFMANN-LA ROCHE INC. (US) 1990-12-04 US claimed
US-4975438-A ANTICOAGULANT HOFFMANN-LA ROCHE INC. (US) 1990-12-04 US disclosed