SCHEMBL10400705

SCHEMBL10400705

COc1cc2cc(C(=O)NO)sc2cc1OC.[NaH]

nearest known ligand 0.78

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 6/20 0.78
HDAC3 O15379 5/20 0.78
HDAC4 P56524 5/20 0.78
HDAC7 Q8WUI4 5/20 0.78
HDAC2 Q92769 5/20 0.78
HDAC10 Q969S8 5/20 0.78
HDAC11 Q96DB2 5/20 0.78
HDAC8 Q9BY41 5/20 0.78
HDAC6 Q9UBN7 5/20 0.78
HDAC9 Q9UKV0 5/20 0.78
HDAC5 Q9UQL6 5/20 0.78
STING1 Q86WV6 13/20 0.58
ACHE P22303 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10400717 0.98 HDAC1 (0.80) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL20049489 0.87 HDAC3 (0.64) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL10400707 0.84 HDAC3 (0.61) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL1590372 0.83 STING1 (0.61) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL1589579 0.81 STING1 (0.68) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL9204578 0.81 STING1 (0.63) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL3060771 0.81 HDAC3 (0.56) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL1590345 0.80 STING1 (0.61) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL7106760 0.80 STING1 (0.61) HDAC1HDAC3HDAC4HDAC7HDAC2
Hydrochloric Acid SCHEMBL4457221 0.79 HDAC3 (0.55) HDAC1HDAC3HDAC4HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4929636-A Positive inotrophic benzothiazole and benzothiophene compositions and method of use therefor AKZO N.V. (NL) 1990-05-29 US disclosed
EP-0158380-B1 BENZOTHIAZOLE AND BENZOTHIOPHENE DERIVATIVES AKZO N.V. (NL) 1989-01-11 EP disclosed
US-4665206-A Benzothiophene derivatives AKZO N.V. (NL) 1987-05-12 US disclosed
EP-0158380-A1 Benzothiazole and benzothiophene derivatives AKZO N.V. (NL) 1985-10-16 EP disclosed