SCHEMBL10401451

SCHEMBL10401451

CCC[n+]1cc(Br)cc(CC(=O)NCCOC(=O)Nc2cccc3ccccc23)c1C(=O)Nc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
HPGD P15428 1/20 0.42
EPHX1 P07099 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
KDM4E B2RXH2 4/20 0.35
MAPT P10636 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 2/20 0.35
KMT2A Q03164 4/20 0.35
MEN1 O00255 3/20 0.35
HTT P42858 2/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MTNR1A P48039 1/20 0.34
GSK3B P49841 1/20 0.34
CDC25B P30305 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10401453 0.83 ALDH1A1 (0.41) ALDH1A1HPGDEPHX1SMN1; SMN2KDM4E
SCHEMBL10401452 0.81 ALDH1A1 (0.41) ALDH1A1HPGDEPHX1NPSR1SMN1; SMN2
Hydrochloric Acid SCHEMBL9524170 0.80 ALDH1A1 (0.41) ALDH1A1HPGDEPHX1NPSR1SMN1; SMN2
Iodide SCHEMBL9525393 0.80 ALDH1A1 (0.41) ALDH1A1HPGDEPHX1NPSR1SMN1; SMN2
Hydrochloric Acid SCHEMBL9524176 0.80 ALDH1A1 (0.42) ALDH1A1HPGDEPHX1KDM4EMAPT
Iodide SCHEMBL9525399 0.80 ALDH1A1 (0.42) ALDH1A1HPGDEPHX1KDM4EMAPT
Hydrochloric Acid SCHEMBL9524106 0.73 ALDH1A1 (0.40) ALDH1A1HPGDEPHX1KMT2AMEN1
SCHEMBL9526051 0.73 MEN1 (0.44) ALDH1A1HPGDNPSR1SMN1; SMN2KDM4E
Hydrochloric Acid SCHEMBL9524164 0.72 ALDH1A1 (0.41) ALDH1A1HPGDEPHX1KDM4EMAPT
Iodide SCHEMBL9525383 0.72 ALDH1A1 (0.41) ALDH1A1HPGDEPHX1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed