SCHEMBL10404129

SCHEMBL10404129

CCOC(=O)c1c(=O)c2c(F)c(F)c(N3CCNCC3)c(F)c2n2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
IDO1 P14902 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
MAPK1 P28482 1/20 0.43
HBB P68871 1/20 0.43
HIF1A Q16665 1/20 0.43
STAT3 P40763 1/20 0.40
KDM4E B2RXH2 5/20 0.40
GAA P10253 3/20 0.40
HPGD P15428 3/20 0.40
GLA P06280 1/20 0.40
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
NPSR1 Q6W5P4 2/20 0.38
RXFP1 Q9HBX9 1/20 0.38
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
APAF1 O14727 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10404626 0.90 ALDH1A1 (0.44) ALDH1A1IDO1CYP1A2CYP3A4MAPK1
SCHEMBL10403241 0.86 DHODH (0.37) ALDH1A1IDO1STAT3KDM4EHPGD
SCHEMBL10385618 0.85 ALDH1A1 (0.52) ALDH1A1IDO1CYP1A2CYP3A4MAPK1
SCHEMBL10404697 0.77 ALDH1A1 (0.49) ALDH1A1IDO1CYP1A2CYP3A4MAPK1
SCHEMBL10777266 0.71 MEN1 (0.55) ALDH1A1CYP1A2MAPK1STAT3KDM4E
SCHEMBL10771130 0.71 NPC1 (0.37) ALDH1A1STAT3GAAMEN1KMT2A
SCHEMBL13312621 0.70 ALDH1A1 (0.62) ALDH1A1MAPK1KDM4EMEN1KMT2A
SCHEMBL14177932 0.69 SMN1; SMN2 (0.49) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL10385637 0.68 ALDH1A1 (0.52) ALDH1A1IDO1CYP1A2CYP3A4MAPK1
SCHEMBL4755207 0.67 RECQL (0.64) ALDH1A1KDM4EMEN1KMT2ARECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4923868-A BACTERICIDES AMERICAN CYANAMID COMPANY (US) 1990-05-08 US claimed