SCHEMBL10409072

SCHEMBL10409072

CCCN(CCC)CCc1ccc(OCc2ccccc2)c(NC=O)c1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.51
EBP Q15125 1/20 0.51
TMEM97 Q5BJF2 1/20 0.51
BCHE P06276 4/20 0.47
DRD2 P14416 1/20 0.47
OPRM1 P35372 1/20 0.47
DRD3 P35462 1/20 0.47
OPRD1 P41143 1/20 0.47
OPRK1 P41145 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10410244 0.91 SIGMAR1 (0.51) SIGMAR1EBPTMEM97BCHEDRD2
SCHEMBL11672572 0.84 BCHE (0.43) BCHEOPRM1OPRD1OPRK1
SCHEMBL10410171 0.83 SIGMAR1 (0.53) SIGMAR1EBPTMEM97DRD2OPRM1
SCHEMBL6812942 0.83 FOLH1 (0.45)
Bromide SCHEMBL10553517 0.82 SIGMAR1 (0.52) SIGMAR1EBPTMEM97DRD2OPRM1
SCHEMBL5665750 0.81 KDM4E (0.38) BCHEDRD2OPRM1DRD3OPRD1
Bromide SCHEMBL10805839 0.81 SIGMAR1 (0.54) SIGMAR1EBPTMEM97BCHEDRD2
SCHEMBL10555893 0.81 SIGMAR1 (0.48) SIGMAR1EBPTMEM97BCHEDRD2
SCHEMBL10410635 0.81 FFAR4 (0.43)
SCHEMBL10409074 0.78 SIGMAR1 (0.57) SIGMAR1EBPTMEM97BCHEDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4958026-A HYPOTENSIVE AGENTS SCHERING AKTIENGESLLSCHAFT (DE) 1990-09-18 US disclosed
EP-0189473-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS. SCHERING AG (DE) 1986-08-06 EP disclosed
US-4598068-A Benzylphenyl osides, method of preparation and use therefor Societe de Recheres Industrielles (FR) 1986-07-01 US disclosed
WO-1986001204-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1986-02-27 WO disclosed