SCHEMBL10409097

SCHEMBL10409097

CN(C)/C=C/c1ccc([N+](=O)[O-])c(OCc2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 4/20 0.47
BACE1 P56817 1/20 0.45
CYP19A1 P11511 3/20 0.45
KDM4E B2RXH2 3/20 0.45
LMNA P02545 2/20 0.45
TLR4 O00206 1/20 0.44
TLR2 O60603 1/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
MAPT P10636 3/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
MYC P01106 1/20 0.43
MAX P61244 1/20 0.43
ALDH1A1 P00352 3/20 0.43
POLB P06746 2/20 0.43
NPC1 O15118 1/20 0.43
USP2 O75604 1/20 0.43
NSD2 O96028 1/20 0.43
HSP90AA1 P07900 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10409098 1.00 APP (0.47) APPBACE1CYP19A1KDM4ELMNA
SCHEMBL8280918 0.84 MAPT (0.49) CYP19A1KDM4ELMNAMAPTMEN1
SCHEMBL9380325 0.82 KDM4E (0.55) APPBACE1CYP19A1KDM4ELMNA
SCHEMBL9380318 0.82 KDM4E (0.55) APPBACE1CYP19A1KDM4ELMNA
SCHEMBL649491 0.82 MAPT (0.55) BACE1LMNAMAOAMAOBMAPT
SCHEMBL9380841 0.82 KDM4E (0.63) APPBACE1KDM4ELMNAALDH1A1
SCHEMBL11842261 0.82 MEN1 (0.46) BACE1CYP19A1LMNAMAPTMEN1
SCHEMBL11842249 0.82 MEN1 (0.46) BACE1CYP19A1LMNAMAPTMEN1
SCHEMBL9380836 0.82 KDM4E (0.63) APPBACE1KDM4ELMNAALDH1A1
SCHEMBL6248370 0.81 BACE1 (0.45) APPBACE1KDM4ELMNATLR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4958026-A HYPOTENSIVE AGENTS SCHERING AKTIENGESLLSCHAFT (DE) 1990-09-18 US disclosed
EP-0189473-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS. SCHERING AG (DE) 1986-08-06 EP disclosed
WO-1986001204-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1986-02-27 WO disclosed