SCHEMBL10423902

SCHEMBL10423902

CCOC(=O)CC(=CC(C)C)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.50
MGAM O43451 1/20 0.50
SI P14410 1/20 0.50
MGAM2 Q2M2H8 1/20 0.50
GRIK1 P39086 2/20 0.44
GRIA2 P42262 2/20 0.44
GRIA4 P48058 2/20 0.44
GRIK3 Q13003 2/20 0.44
GRIK5 Q16478 2/20 0.44
GRIA1 P42261 1/20 0.44
GRIK2 Q13002 1/20 0.44
ALDH1A1 P00352 3/20 0.38
TRPA1 O75762 1/20 0.38
LMNA P02545 1/20 0.36
HCAR2 Q8TDS4 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NLRP3 Q96P20 1/20 0.34
CYP2D6 P10635 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4661591 0.85 GAA (0.50) GAAMGAMSIMGAM2GRIK1
SCHEMBL30904961 0.82 GRIK1 (0.48) GAAMGAMSIMGAM2GRIK1
SCHEMBL10382305 0.82 GRIK1 (0.48) GAAMGAMSIMGAM2GRIK1
SCHEMBL27781924 0.80 GAA (0.58) GAAMGAMSIMGAM2GRIK1
SCHEMBL28601595 0.77 GAA (0.54) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL13293249 0.77 GAA (0.54) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL3504490 0.77 GAA (0.54) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL5879637 0.77 GAA (0.54) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL14349108 0.76 GRIK1 (0.43) GAAGRIK1GRIA2GRIA4GRIK3
SCHEMBL2637977 0.76 NR1H4 (0.45) ALDH1A1LMNAL3MBTL1SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4918105-A Novel compounds with collagenase-inhibiting activity, a process for their preparation and pharmaceutical compositions in which these compounds are present SA LABORATOIRE ROGER BELLON (FR) 1990-04-17 US disclosed