SCHEMBL10423960

SCHEMBL10423960

COc1ccc(C2(Oc3c(F)c(F)c(F)c(F)c3F)CCN(C)CC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
SLC6A4 P31645 2/20 0.38
KMT2A Q03164 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A3 Q01959 1/20 0.37
MMP1 P03956 1/20 0.37
MMP9 P14780 1/20 0.37
MMP13 P45452 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MAOB P27338 2/20 0.36
NPC1 O15118 1/20 0.36
PKM P14618 1/20 0.36
PKLR P30613 1/20 0.36
RAB9A P51151 1/20 0.36
MAOA P21397 1/20 0.36
CHRM5 P08912 2/20 0.36
CHRM3 P20309 2/20 0.36
CHRM1 P11229 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10423408 0.99 GRIN1 (0.38) GRIN1GRIN2AGRIN2BSLC6A4KMT2A
SCHEMBL10423359 0.87 OPRM1 (0.44) SLC6A4KMT2ASLC6A3MMP13
Hydrochloric Acid SCHEMBL10423965 0.85 OPRM1 (0.46) SLC6A4KMT2ASLC6A3MMP13
Hydrochloric Acid SCHEMBL10424433 0.84 OPRM1 (0.47) KMT2ASLC6A3
SCHEMBL10423994 0.84 OPRM1 (0.46) SLC6A4KMT2A
SCHEMBL10423987 0.84 OPRM1 (0.44) SLC6A4
SCHEMBL10423409 0.82 PDE2A (0.42) SLC6A4
Oxalic Acid SCHEMBL10423990 0.78 OPRM1 (0.45) SLC6A4KMT2ACHRM5CHRM3CHRM1
Fumaric Acid SCHEMBL10458883 0.75 OPRM1 (0.43) KMT2A
Fumaric Acid SCHEMBL10423357 0.75 OPRM1 (0.43) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4954511-A ALLEVIATING PAIN, TREATING DEPRESSION, CONVULSIONS AND HYPERTENSION HOECHST-ROUSSELL PHARMACEUTICALS INC. (US) 1990-09-04 US claimed
US-4954511-A ALLEVIATING PAIN, TREATING DEPRESSION, CONVULSIONS AND HYPERTENSION HOECHST-ROUSSELL PHARMACEUTICALS INC. (US) 1990-09-04 US disclosed
US-4914204-A ANALGESICS, ANTIDEPRESSANTS, ANTICONVULSANTS, HYPOTENSIVE AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1990-04-03 US disclosed
EP-0333027-A1 4-Pentafluorophenoxypiperidines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-09-20 EP disclosed