SCHEMBL10424596

SCHEMBL10424596

O=C(O)CSc1ccccc1CC(=O)O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.59
HPGD P15428 2/20 0.54
CYP2C9 P11712 2/20 0.54
CYP2C19 P33261 1/20 0.54
AKR1B1 P15121 2/20 0.53
FFAR1 O14842 1/20 0.53
TDP1 Q9NUW8 1/20 0.52
KDM4E B2RXH2 3/20 0.50
ALDH1A1 P00352 1/20 0.50
HSD17B10 Q99714 1/20 0.50
MMP2 P08253 1/20 0.47
MMP9 P14780 1/20 0.47
MMP12 P39900 1/20 0.47
CDC25B P30305 1/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
GAA P10253 1/20 0.44
APEX1 P27695 1/20 0.43
PAM P19021 1/20 0.43
AKR1B10 O60218 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL670712 0.87 HPGD (0.50) CYP1A2HPGDCYP2C9CYP2C19AKR1B1
SCHEMBL21328440 0.85 CYP1A2 (0.59) CYP1A2HPGDCYP2C9FFAR1KDM4E
SCHEMBL14273063 0.83 CYP1A2 (0.73) CYP1A2HPGDCYP2C9FFAR1KDM4E
SCHEMBL8631418 0.83 POLB (0.53) HPGDCYP2C9CYP2C19AKR1B1TDP1
SCHEMBL11533963 0.83 CYP1A2 (0.58) CYP1A2HPGDCYP2C9CYP2C19FFAR1
SCHEMBL4828911 0.82 AKR1B1 (0.59) CYP1A2HPGDCYP2C9CYP2C19AKR1B1
SCHEMBL4438683 0.82 CYP2C9 (0.69) HPGDCYP2C9CYP2C19AKR1B1TDP1
SCHEMBL14273050 0.80 CYP1A2 (0.54) CYP1A2HPGDCYP2C9FFAR1KDM4E
SCHEMBL711355 0.78 CYP2C9 (0.56) HPGDCYP2C9CYP2C19AKR1B1TDP1
SCHEMBL4832670 0.78 CYP2C9 (0.56) CYP1A2HPGDCYP2C9CYP2C19AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4935441-A Flavene and thioflavene derivates, processes for their manufacture, pharmaceutical preparations that contain such compounds, and the use of the latter ZYMA SA (CH) 1990-06-19 US disclosed
EP-0139615-B1 FLAVENE AND THIOFLAVENE DERIVATIVES, PROCESSES FOR THEIR MANUFACTURE, PHARMACEUTICAL PREPARATIONS THAT CONTAIN SUCH COMPOUNDS, AND THE USE OF THE LATTER Zyma SA (CH) 1989-04-19 EP disclosed
EP-0139615-A2 Flavene and thioflavene derivatives, processes for their manufacture, pharmaceutical preparations that contain such compounds, and the use of the latter Zyma SA (CH) 1985-05-02 EP disclosed