SCHEMBL10429347

SCHEMBL10429347

O=C(Nc1ccc(-c2nsc3c(=O)[nH]nnc23)cc1)OCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.50
POLB P06746 1/20 0.46
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
MGLL Q99685 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KDM1A O60341 2/20 0.41
MAOA P21397 2/20 0.41
MAOB P27338 2/20 0.41
RCOR1 Q9UKL0 1/20 0.41
ENPP2 Q13822 1/20 0.40
PTPN1 P18031 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10429313 0.72 NOTUM (0.38) POLBTP53MAPTSMN1; SMN2PTGDR2
SCHEMBL10429372 0.72 ROCK2 (0.52) ROCK2POLBPDE3BPDE3ATP53
SCHEMBL11114283 0.70 PDGFRB (0.55) ROCK2POLBPDE3BPDE3ATP53
SCHEMBL10429350 0.70 KDR (0.36) PDE3BPDE3AALDH1A1
SCHEMBL9128045 0.69 ROCK2 (0.69) ROCK2POLBPDE3BPDE3ATP53
SCHEMBL11119482 0.69 ROCK2 (0.62) ROCK2POLBPDE3BPDE3ATP53
Benzyl Phenylcarbamate SCHEMBL1222943 0.69 POLB (0.78) ROCK2POLBTP53MAPTMGLL
SCHEMBL10259763 0.69 POLB (0.83) ROCK2POLBPDE3BPDE3ATP53
SCHEMBL7297495 0.68 ROCK2 (0.57) ROCK2POLBPDE3BPDE3ATP53
SCHEMBL7295061 0.68 ROCK2 (0.60) ROCK2POLBPDE3BPDE3ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274654-A2 1,2,3-Triazin-4(3H)-one derivatives, process for their preparation and medicaments containing them F. HOFFMANN-LA ROCHE AG (CH) 1988-07-20 EP claimed
US-4920119-A XANTHINE OXIDASE INHIBITORS; CONTROL OR PREVENTION OF GOUT OR ISCHEMIA HOFFMANN-LA ROCHE INC. (US) 1990-04-24 US disclosed
EP-0296374-A2 Glycosylated aminoacids and peptides HOECHST AKTIENGESELLSCHAFT (DE) 1988-12-28 EP disclosed
EP-0274654-A2 1,2,3-Triazin-4(3H)-one derivatives, process for their preparation and medicaments containing them F. HOFFMANN-LA ROCHE AG (CH) 1988-07-20 EP disclosed