SCHEMBL10440288

SCHEMBL10440288

C[C@H](O)[C@H]1C(=O)N2C(C(=O)O)=C(SCc3ccccc3)[C@H](C)[C@H]12

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.48
PTGS1 P23219 1/20 0.48
PDE4A P27815 1/20 0.48
CACNA1C Q13936 1/20 0.46
ELANE P08246 7/20 0.42
ABCC2 Q92887 1/20 0.41
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
FAP Q12884 1/20 0.35
KDM6B O15054 1/20 0.34
KDM4A O75164 1/20 0.34
KDM4D Q6B0I6 1/20 0.34
HIF1AN Q9NWT6 1/20 0.34
KDM5B Q9UGL1 1/20 0.34
KDM2A Q9Y2K7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21081301 1.00 ESR1 (0.48) ESR1PTGS1PDE4ACACNA1CELANE
SCHEMBL9696446 0.91 ESR1 (0.45) ESR1PTGS1PDE4ACACNA1CELANE
SCHEMBL10440510 0.90 CACNA1C (0.40) ESR1PTGS1PDE4ACACNA1CELANE
SCHEMBL21081300 0.90 ESR1 (0.47) ESR1PTGS1PDE4ACACNA1CELANE
SCHEMBL9696350 0.85 ESR1 (0.47) ESR1PTGS1PDE4ACACNA1CELANE
SCHEMBL10440442 0.85 ESR1 (0.44) ESR1PTGS1PDE4ACACNA1CELANE
SCHEMBL10682791 0.84 ESR1 (0.44) ESR1PTGS1PDE4ACACNA1CELANE
SCHEMBL10683098 0.84 ESR1 (0.43) ESR1PTGS1PDE4ACACNA1CELANE
SCHEMBL10683095 0.84 ESR1 (0.43) ESR1PTGS1PDE4ACACNA1CELANE
SCHEMBL10440528 0.83 CACNA1C (0.51) ESR1PTGS1PDE4ACACNA1CELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0372582-A2 6-Aminoalkyl carbapenems Bristol-Myers Squibb Company (US) 1990-06-13 EP disclosed