SCHEMBL10683098

SCHEMBL10683098

Cc1cc(CSC2=C(C(=O)O)N3C(=O)[C@H]([C@@H](C)O)[C@@H]3[C@H]2C)ccn1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.43
PTGS1 P23219 1/20 0.43
PDE4A P27815 1/20 0.43
CACNA1C Q13936 1/20 0.42
ABCC2 Q92887 1/20 0.37
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
FAP Q12884 1/20 0.33
ELANE P08246 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10683095 1.00 ESR1 (0.43) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL10682791 0.85 ESR1 (0.44) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL21081301 0.84 ESR1 (0.48) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL10440288 0.84 ESR1 (0.48) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL10679749 0.82 CACNA1C (0.42) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL10679752 0.82 CACNA1C (0.42) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL10440442 0.80 ESR1 (0.44) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL10683072 0.80 KDM4E (0.53) ESR1PTGS1PDE4AKDM4ELMNA
SCHEMBL10683068 0.80 KDM4E (0.53) ESR1PTGS1PDE4AKDM4ELMNA
SCHEMBL10679836 0.79 ESR1 (0.43) ESR1PTGS1PDE4ACACNA1CABCC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4746736-A THIENAMYCINS, BACTERICIDES BRISTOL-MYERS COMPANY (US) 1988-05-24 US disclosed
US-4732977-A BACTERICIDES BRISTOL MYERS COMPANY (US) 1988-03-22 US disclosed
US-4644061-A Carbapenem antibiotics BRISTOL-MYERS COMPANY (US) 1987-02-17 US disclosed