SCHEMBL10450802

SCHEMBL10450802

CC(C)(C)[Si](C)(C)Oc1ccc(C2CCc3cc(O[Si](C)(C)C(C)(C)C)ccc3C2=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.43
CA1 P00915 4/20 0.43
CA9 Q16790 4/20 0.43
PREP P48147 2/20 0.41
CYP19A1 P11511 3/20 0.41
CYP24A1 Q07973 6/20 0.38
CYP27A1 Q02318 3/20 0.38
CYP26A1 O43174 3/20 0.37
THRA P10827 1/20 0.35
THRB P10828 1/20 0.35
ALOX15 P16050 1/20 0.34
ALOX12 P18054 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9419768 0.84 CA12 (0.43) CA12CA1CA9PREPCYP19A1
SCHEMBL12852985 0.81 CYP19A1 (0.48) CA12CA1CA9PREPCYP19A1
SCHEMBL10042955 0.79 CYP19A1 (0.58) CA12CA1CA9PREPCYP19A1
SCHEMBL6669546 0.78 CYP24A1 (0.53) CYP19A1CYP24A1CYP27A1CYP26A1ALOX15
SCHEMBL24529065 0.76 MAOB (0.48) CA12CA1CA9PREP
SCHEMBL30598686 0.74 CYP26A1 (0.59) CYP19A1CYP24A1CYP27A1CYP26A1THRA
SCHEMBL20798296 0.74 CYP26A1 (0.59) CYP19A1CYP24A1CYP27A1CYP26A1THRA
SCHEMBL6113027 0.74 MAOB (0.50) CA12CA1CA9PREP
SCHEMBL5405281 0.74 MAOB (0.50) CA12CA1CA9PREP
SCHEMBL15965361 0.74 CYP19A1 (0.62) PREPCYP19A1ALOX15ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4904661-A ANTIESTROGENS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-02-27 US disclosed
US-4732912-A ANTIESTROGENS, ANTITUMOR AGENTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-03-22 US disclosed
EP-0124369-A1 Phenol derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-11-07 EP disclosed