SCHEMBL10461663

SCHEMBL10461663

OC(c1cccc(F)c1)(c1cccc(F)c1)C(c1ccccc1)N1CCCCC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 11/20 0.60
KCNH2 Q12809 9/20 0.60
CYP3A4 P08684 5/20 0.55
CYP2D6 P10635 5/20 0.55
CYP2C9 P11712 5/20 0.55
CYP2C19 P33261 5/20 0.55
HTT P42858 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
CHRNB2 P17787 1/20 0.43
SLC6A2 P23975 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA4 P43681 1/20 0.43
SLC6A3 Q01959 1/20 0.43
CYP1A2 P05177 4/20 0.42
KCNE1 P15382 1/20 0.42
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
OPRL1 P41146 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480997 0.85 KCNA5 (0.73) KCNA5KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL12587918 0.85 KCNA5 (0.73) KCNA5KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL480998 0.85 KCNA5 (0.73) KCNA5KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL5541536 0.85 KCNA5 (0.73) KCNA5KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL13649151 0.83 KCNA5 (0.73) KCNA5KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL1242816 0.78 KCNA5 (0.73) KCNA5KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL1243260 0.75 KCNA5 (1.00) KCNA5KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL1241166 0.74 KCNA5 (0.81) KCNA5KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL1242084 0.73 KCNA5 (1.00) KCNA5KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL1242863 0.72 KCNA5 (0.81) KCNA5KCNH2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4950674-A Arylalkylheterocyclic amines,N-substituted by aryloxyalkyl group in a method for allergy treatment A. H. ROBINS COMPANY, INCORPORATED (US) 1990-08-21 US disclosed