SCHEMBL10470684

SCHEMBL10470684

O=C(NCc1ccccc1)[C@@H]1CSCN1C(=O)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.46
HTR1B P28222 1/20 0.46
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
HTR2B P41595 1/20 0.46
VHL P40337 1/20 0.46
AADAT Q8N5Z0 1/20 0.46
ALDH1A1 P00352 2/20 0.46
USP2 O75604 1/20 0.46
HPGD P15428 1/20 0.46
MC4R P32245 1/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
PKM P14618 1/20 0.45
CYP2C19 P33261 1/20 0.45
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10470346 0.81 EPHX2 (0.56)
SCHEMBL10340335 0.79 ACE (0.44) ALDH1A1HPGDCA2TSHR
SCHEMBL3750871 0.79 ACE (0.44) ALDH1A1HPGDCA2TSHR
SCHEMBL10716752 0.78 HTR1A (0.45) HTR1AHTR1BHTR2AHTR2CHTR2B
SCHEMBL10716748 0.78 HTR1A (0.45) HTR1AHTR1BHTR2AHTR2CHTR2B
SCHEMBL10340448 0.75 RECQL (0.48) ALDH1A1USP2HPGDPKM
SCHEMBL10340422 0.75 RECQL (0.48) ALDH1A1USP2HPGDPKM
SCHEMBL30090978 0.75 RECQL (0.48) ALDH1A1USP2HPGDPKM
SCHEMBL10340322 0.75 RECQL (0.48) ALDH1A1USP2HPGDPKM
SCHEMBL10340323 0.75 RECQL (0.48) ALDH1A1USP2HPGDPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4904680-A IMMUNOLOGY SANKYO COMPANY, LIMITED (JP) 1990-02-27 US claimed
EP-0173441-A1 Amino acid derivatives having anti-tumor activity and compositions containing them SANKYO COMPANY LIMITED (JP) 1986-03-05 EP claimed
US-4904680-A IMMUNOLOGY SANKYO COMPANY, LIMITED (JP) 1990-02-27 US disclosed
EP-0173441-A1 Amino acid derivatives having anti-tumor activity and compositions containing them SANKYO COMPANY LIMITED (JP) 1986-03-05 EP disclosed