SCHEMBL10474240

SCHEMBL10474240

NC(=O)c1ncn2c(-c3cccc(Cl)c3)ccnc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.44
BACE1 P56817 1/20 0.43
NUDT1 P36639 1/20 0.43
NR3C2 P08235 1/20 0.42
TLR8 Q9NR97 1/20 0.42
KMO O15229 1/20 0.40
KDM4E B2RXH2 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
JAK2 O60674 1/20 0.39
DYRK1B Q9Y463 2/20 0.39
MAP2K1 Q02750 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
NTRK1 P04629 2/20 0.39
PIM1 P11309 2/20 0.39
ACVR1 Q04771 1/20 0.39
FGFR3 P22607 1/20 0.38
KDR P35968 1/20 0.38
GAA P10253 1/20 0.38
IDO1 P14902 1/20 0.38
PARP1 P09874 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10474901 0.84 NTRK1 (0.53) IKBKBNR3C2KDM4EDYRK1BMAP2K1
SCHEMBL10473295 0.84 CLK4 (0.53) IKBKBTLR8KDM4EKDM4CDYRK1B
SCHEMBL10473059 0.84 KMO (0.43) NR3C2TLR8KMOKDM4EKDM4C
SCHEMBL10473420 0.82 MAPT (0.47) IKBKBTLR8KDM4EJAK2CLK4
SCHEMBL10473172 0.82 KDM4E (0.61) TLR8KMOKDM4EDYRK1BPARP1
SCHEMBL10474874 0.81 TSHR (0.43) TLR8KDM4EGAANPC1RAB9A
SCHEMBL10474226 0.80 EGLN2 (0.42) BACE1KDM4EKDM4CJAK2NTRK1
SCHEMBL10473249 0.80 MKNK1 (0.52) IKBKBTLR8KDM4EDYRK1BMAP2K1
SCHEMBL10473048 0.77 MAPT (0.45) JAK2NTRK1PIM1KDR
SCHEMBL10475196 0.76 NTRK1 (0.55) IKBKBNR3C2TLR8KDM4CDYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4904658-A Substituted-6H,8H-pyrimido-[1,2,3-cd]purine-8,10-(9H)-diones and substituted-6H,10H-pyrimido[1,2-cd]purin-10-ones AMERICAN CYANAMID COMPANY (US) 1990-02-27 US disclosed
US-4888345-A HYPOTENSIVE AND ANXIOLYTIC AGENTS; CHEMICAL INTERMEDIATES AMERICAN CYANAMID COMPANY (US) 1989-12-19 US disclosed