SCHEMBL10476263

SCHEMBL10476263

CC(NC(=O)c1ccc(CSc2c(Cl)ccc3c2CCNCC3)cc1)C1CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 5/20 0.43
SMYD3 Q9H7B4 2/20 0.39
MCHR1 Q99705 1/20 0.38
P2RX7 Q99572 2/20 0.37
PPARG P37231 1/20 0.36
CNR1 P21554 2/20 0.36
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
MAPK14 Q16539 2/20 0.36
PDE6D O43924 1/20 0.36
ACKR3 P25106 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10476296 1.00 CNR2 (0.43) CNR2SMYD3MCHR1P2RX7PPARG
SCHEMBL10476261 1.00 CNR2 (0.43) CNR2SMYD3MCHR1P2RX7PPARG
Succinic Acid SCHEMBL507022 0.96 CNR2 (0.41) CNR2SMYD3MCHR1P2RX7PPARG
Succinic Acid SCHEMBL507228 0.96 CNR2 (0.41) CNR2SMYD3MCHR1P2RX7PPARG
SCHEMBL10274759 0.86 RXFP1 (0.44) PDE6D
SCHEMBL10476151 0.83 HDAC6 (0.42) SMYD3P2RX7MAPK14
Succinic Acid SCHEMBL507841 0.82 RXFP1 (0.43) PDE6D
Hydrochloric Acid SCHEMBL2369279 0.82 HDAC6 (0.41) SMYD3P2RX7MAPK14
SCHEMBL10476175 0.82 ALDH1A1 (0.41) MCHR1
SCHEMBL10476173 0.82 ALDH1A1 (0.41) MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8580780-B2 6 substituted 2, 3,4,5 tetrahydro-1H-benzo[d]azepines as 5-HT2C receptor agonist ELI LILLY AND COMPANY (US) 2013-11-12 US claimed
EP-2479168-A1 6-Substituted 2,3,4,5-Tetrahydro-1H-Benzo [d]Azepines as 5-HT2C Receptor Agonists ELI LILLY AND COMPANY (US) 2012-07-25 EP claimed