SCHEMBL10476629

SCHEMBL10476629

Cc1ccc(-c2noc([C@@H](C)OC3CCN(c4nc(C(C)C)no4)CC3)n2)cc1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 14/20 0.47
MAPT P10636 3/20 0.43
LMNA P02545 2/20 0.43
GPR183 P32249 1/20 0.40
ALOX5AP P20292 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4113153 0.91 GPR119 (0.48) GPR119MAPTLMNAGPR183ALOX5AP
SCHEMBL4102142 0.89 GPR119 (0.45) GPR119MAPTLMNAGPR183ALOX5AP
SCHEMBL4095100 0.88 GPR119 (0.55) GPR119MAPTLMNAGPR183
SCHEMBL4106749 0.87 GPR119 (0.44) GPR119MAPTLMNAGPR183
SCHEMBL4114745 0.85 GPR119 (0.43) GPR119MAPTLMNAGPR183
SCHEMBL4114736 0.84 GPR119 (0.55) GPR119GPR183
SCHEMBL4101235 0.83 GPR119 (0.50) GPR119
SCHEMBL4112505 0.81 GPR119 (0.67) GPR119
SCHEMBL10476580 0.81 GPR119 (0.43) GPR119MAPTLMNAGPR183ALOX5AP
SCHEMBL14403714 0.73 GPR119 (0.57) GPR119MAPTLMNAGPR183

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013201-B1 HETEROCYCLIC GPCR AGONISTS PROSIDION LTD (GB) 2012-07-25 EP claimed