SCHEMBL10477117

SCHEMBL10477117

c1ccc2c(c1)CC1CNCCC2C1

nearest known ligand 0.73

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 8/20 0.73
CHRNA4 P43681 8/20 0.73
CHRNA7 P36544 3/20 0.45
CHRNB4 P30926 2/20 0.45
CHRNA3 P32297 2/20 0.45
KDM1A O60341 2/20 0.43
KDM1B Q8NB78 1/20 0.43
HTR2C P28335 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5994733 0.84 CHRNB2 (1.00) CHRNB2CHRNA4CHRNA7CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL7137773 0.83 CHRNB2 (0.96) CHRNB2CHRNA4CHRNA7CHRNB4CHRNA3
SCHEMBL11705873 0.78 CHRNB2 (0.59) CHRNB2CHRNA4KDM1A
SCHEMBL32674546 0.76 CHRNB2 (0.66) CHRNB2CHRNA4KDM1A
SCHEMBL11699947 0.75 CHRNB2 (0.56) CHRNB2CHRNA4HTR2C
SCHEMBL6545918 0.75 CHRNB2 (0.56) CHRNB2CHRNA4HTR2C
SCHEMBL11538560 0.74 CHRNB4 (0.72) CHRNB2CHRNA4CHRNB4CHRNA3HTR2C
SCHEMBL11703659 0.74 CHRNB2 (0.54) CHRNB2CHRNA4HTR2C
SCHEMBL11703811 0.74 CHRNB2 (0.54) CHRNB2CHRNA4HTR2C
Hydrochloric Acid SCHEMBL11543466 0.73 CHRNB4 (0.69) CHRNB2CHRNA4CHRNB4CHRNA3HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1020103-C 2,3,4,5,6,7-hexahydro-2,7-methylene-1,5-benzoxazonin and 1,4-benzoxazonin MADAUS & CO DR (DE) 1993-03-17 CN disclosed
US-4859664-A Derivatives of 2,3,4,5,6,7-hexahydro-2,7-methano-1,5-benzoxazonines and -1,4-benzoxazonines, processes for their production and their use as pharmaceuticals MADAUS GMBH & COMPANY (DE) 1989-08-22 US disclosed
CN-87106267-A 2, 3, 4, 5, 6, 7-hexahydro-2, 7-methano-1, 5-benzoxazonin and-1, 4-benzoxazonin, process for their preparation and pharmaceutical compositions containing them 1988-04-13 CN disclosed
US-4082744-A CNS, ANALGESICS, ANTITUSSIVE, SEDATIVES NIHON IYAKUHIN KOGYO CO., LTD. (JA) 1978-04-04 US disclosed
US-4008219-A CNS ANALGESIC, ANTITUSSIVE, SEDATIVE NIHON IYAKUHIN KOGYO CO., LTD. (JA) 1977-02-15 US disclosed