SCHEMBL10482964

SCHEMBL10482964

CN(C(=N)N)C1CCN(c2nc3ccccc3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.76

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 19/20 0.76
CYP2D6 P10635 17/20 0.76
KCNH2 Q12809 11/20 0.76
CHRM1 P11229 8/20 0.71
ADRA2A P08913 1/20 0.61
HTR2B P41595 1/20 0.61
PDE4D Q08499 1/20 0.61
PDE3A Q14432 1/20 0.61
HTR3A P46098 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL10529808 0.95 HRH1 (0.69) HRH1CYP2D6KCNH2CHRM1ADRA2A
SCHEMBL10527191 0.89 HRH1 (0.73) HRH1CYP2D6KCNH2CHRM1ADRA2A
SCHEMBL10527187 0.89 HRH1 (0.73) HRH1CYP2D6KCNH2CHRM1ADRA2A
SCHEMBL10527217 0.87 HRH1 (0.68) HRH1CYP2D6KCNH2CHRM1ADRA2A
SCHEMBL10483537 0.87 HRH1 (0.80) HRH1CYP2D6KCNH2CHRM1ADRA2A
SCHEMBL10529818 0.86 HRH1 (0.66) HRH1CYP2D6KCNH2CHRM1ADRA2A
SCHEMBL10527210 0.85 HRH1 (0.68) HRH1CYP2D6KCNH2CHRM1ADRA2A
SCHEMBL10529977 0.85 HRH1 (0.73) HRH1CYP2D6KCNH2CHRM1ADRA2A
SCHEMBL10338043 0.83 HRH1 (0.71) HRH1CYP2D6KCNH2CHRM1ADRA2A
SCHEMBL10337872 0.82 HRH1 (0.71) HRH1CYP2D6KCNH2CHRM1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-1034978-A None JP disclosed
US-4857536-A Antihistaminic benzimidazole derivatives SYNTHELABO (FR) 1989-08-15 US disclosed