SCHEMBL10488253

SCHEMBL10488253

CCCCC1c2ccccc2C(=O)c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.44
ACHE P22303 1/20 0.44
ALDH1A1 P00352 2/20 0.43
CYP3A4 P08684 2/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
MAPK1 P28482 1/20 0.43
CYP2C19 P33261 1/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
PTGS1 P23219 1/20 0.43
RAB9A P51151 1/20 0.43
NAPRT Q6XQN6 1/20 0.43
EDNRB P24530 1/20 0.42
EDNRA P25101 1/20 0.42
MEN1 O00255 1/20 0.41
CDC25B P30305 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL313685 0.88 ACHE (0.55) BCHEACHECYP3A4LMNATP53
SCHEMBL6903762 0.82 CDC25B (0.46) BCHEALDH1A1CYP3A4LMNACYP1A2
SCHEMBL877438 0.82 HTR2A (0.56) BCHEACHE
SCHEMBL6061696 0.80 HTR2A (0.54) BCHEACHE
SCHEMBL1449246 0.80 HTR2A (0.54) BCHEACHE
SCHEMBL6060774 0.80 HTR2A (0.54) BCHEACHE
SCHEMBL3977109 0.80 HTR2A (0.54) BCHEACHE
SCHEMBL6061312 0.80 HTR2A (0.54) BCHEACHE
SCHEMBL407781 0.80 HTR2A (0.54) BCHEACHE
SCHEMBL6060915 0.80 HTR2A (0.54) BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4803226-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1989-02-07 US disclosed
US-4803221-A Anthracene derivatives BURROUGHS WELLCOME CO. (US) 1989-02-07 US disclosed
EP-0125701-B1 POLYCYCLIC AROMATIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1988-08-03 EP disclosed
US-4719047-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed
US-4719049-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed
EP-0125701-A2 Polycyclic aromatic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-21 EP disclosed