SCHEMBL10488284

SCHEMBL10488284

CC(CO)(CO)NCc1c2ccccc2c(Br)c2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
SLC2A1 P11166 1/20 0.38
CD274 Q9NZQ7 1/20 0.36
NPBWR1 P48145 1/20 0.33
KMT2A Q03164 1/20 0.33
MCHR1 Q99705 1/20 0.33
CCR5 P51681 1/20 0.32
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10488233 0.98 CYP1A2 (0.37) CYP1A2SLC2A1CD274NPBWR1KMT2A
SCHEMBL10488213 0.86 CYP1A2 (0.40) CYP1A2SLC2A1CD274NPBWR1KMT2A
SCHEMBL10488212 0.85 CYP1A2 (0.37) CYP1A2SLC2A1CD274NPBWR1KMT2A
SCHEMBL10488852 0.85 CD274 (0.42) CYP1A2SLC2A1CD274NPBWR1KMT2A
Hydrochloric Acid SCHEMBL10571382 0.85 CYP1A2 (0.39) CYP1A2SLC2A1CD274NPBWR1KMT2A
Hydrochloric Acid SCHEMBL10488854 0.84 NPBWR1 (0.37) CYP1A2SLC2A1CD274NPBWR1KMT2A
SCHEMBL10488837 0.83 KMT2A (0.38) CYP1A2SLC2A1CD274NPBWR1KMT2A
Hydrochloric Acid SCHEMBL10570896 0.83 CD274 (0.41) CYP1A2SLC2A1CD274NPBWR1KMT2A
SCHEMBL10488886 0.83 KDM4E (0.40) CYP1A2SLC2A1CD274LMNAGAA
Hydrochloric Acid SCHEMBL10488883 0.82 KMT2A (0.40) CYP1A2SLC2A1CD274NPBWR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0125702-B1 POLYCYCLIC AROMATIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1987-08-12 EP claimed
EP-0125702-A2 Polycyclic aromatic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-21 EP claimed
US-4803226-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1989-02-07 US disclosed
US-4803221-A Anthracene derivatives BURROUGHS WELLCOME CO. (US) 1989-02-07 US disclosed
US-4719047-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed
US-4719049-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed
EP-0125702-A2 Polycyclic aromatic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-21 EP disclosed