SCHEMBL10488409

SCHEMBL10488409

COC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1ccc(O)c([N+](=O)[O-])c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 4/20 0.60
KMT2A Q03164 4/20 0.60
CYP1A2 P05177 4/20 0.60
ADORA3 P0DMS8 4/20 0.60
CYP3A4 P08684 3/20 0.60
MAPT P10636 3/20 0.60
CYP2C9 P11712 3/20 0.60
CYP2C19 P33261 3/20 0.60
TSHR P16473 3/20 0.60
LMNA P02545 3/20 0.60
CACNA1F O60840 3/20 0.60
CACNA1D Q01668 3/20 0.60
CACNA1S Q13698 3/20 0.60
CACNA1C Q13936 3/20 0.60
CYP2D6 P10635 2/20 0.60
NFKB1 P19838 2/20 0.60
MAPK1 P28482 2/20 0.60
THPO P40225 2/20 0.60
KDM4E B2RXH2 2/20 0.60
ALDH1A1 P00352 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11784675 0.86 KMT2A (0.69) HIF1AKMT2ACYP1A2ADORA3CYP3A4
SCHEMBL27869994 0.82 KMT2A (0.55) HIF1AKMT2ACYP1A2ADORA3CYP3A4
SCHEMBL11860028 0.82 KMT2A (0.65) HIF1AKMT2ACYP1A2ADORA3CYP3A4
SCHEMBL11784686 0.82 KMT2A (0.65) HIF1AKMT2ACYP1A2ADORA3CYP3A4
SCHEMBL8512764 0.82 KMT2A (0.54) HIF1AKMT2ACYP1A2ADORA3CYP3A4
SCHEMBL7160123 0.80 ADORA3 (0.85) HIF1AKMT2ACYP1A2ADORA3CYP3A4
SCHEMBL10692954 0.80 ADORA3 (0.53) HIF1AKMT2ACYP1A2ADORA3CYP3A4
SCHEMBL7882494 0.79 TSHR (0.57) KMT2AADORA3MAPTTSHRCACNA1F
SCHEMBL7885521 0.79 TSHR (0.57) KMT2AADORA3MAPTTSHRLMNA
SCHEMBL30648615 0.79 HIF1A (0.87) HIF1AKMT2ACYP1A2ADORA3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4873254-A ADRENERGIC BLOCKING AGENTS OR CALCIUM CHANNEL BLOCKERS; HYPOTENSIVE AGENTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-10-10 US disclosed