SCHEMBL10488592

SCHEMBL10488592

CSc1cccc(Nc2n[nH]c(C)c2C(=O)O)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.47
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
MAPT P10636 4/20 0.47
POLB P06746 2/20 0.47
TP53 P04637 1/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47
NPC1 O15118 4/20 0.45
RAB9A P51151 4/20 0.45
ABCG2 Q9UNQ0 3/20 0.44
ABCC1 P33527 1/20 0.44
TGFBR1 P36897 1/20 0.43
HPGD P15428 2/20 0.43
ALDH1A1 P00352 2/20 0.43
STAT1 P42224 1/20 0.43
GRM4 Q14833 1/20 0.41
ALPG P10696 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10488620 0.85 SMN1; SMN2 (0.54) SMN1; SMN2MEN1KMT2AMAPTPOLB
SCHEMBL10488953 0.82 MAPT (0.56) SMN1; SMN2MAPTPOLBMAPK1NPC1
SCHEMBL10488935 0.82 EGFR (0.54) SMN1; SMN2MEN1KMT2AMAPK1NPC1
SCHEMBL10488481 0.76 MAPT (0.46) SMN1; SMN2MEN1KMT2AMAPTPOLB
SCHEMBL10488911 0.74 SMN1; SMN2 (0.42) SMN1; SMN2MEN1KMT2AMAPTPOLB
SCHEMBL10488476 0.73 LRRK2 (0.50) SMN1; SMN2MEN1KMT2AMAPTMAPK1
SCHEMBL11085536 0.73 MAPT (0.55) SMN1; SMN2MAPTPOLBMAPK1NPC1
SCHEMBL10488575 0.72 FTO (0.44) SMN1; SMN2ALDH1A1
SCHEMBL5256676 0.72 MEN1 (0.65) SMN1; SMN2MEN1KMT2AMAPTPOLB
SCHEMBL10488610 0.71 CLCN2 (0.47) SMN1; SMN2MAPTPOLBCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4871737-A 3-Amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants muscle relaxants and anxiolytics A. H. ROBINS COMPANY, INCORPORATED (US) 1989-10-03 US disclosed
EP-0315433-A2 3-amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants, muscle relaxants and anxiolytics A.H. ROBINS COMPANY, INCORPORATED (US) 1989-05-10 EP disclosed
US-4826866-A 3-amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants, muscle relaxants and anxiolytics A. H. ROBINS COMPANY, INCORPORATED (US) 1989-05-02 US disclosed