SCHEMBL10488604

SCHEMBL10488604

CCCNc1n[nH]c(C)c1C(=O)OCC

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.65
PDE4D Q08499 1/20 0.61
AURKA O14965 3/20 0.49
MAPT P10636 3/20 0.48
POLB P06746 2/20 0.48
KDM4E B2RXH2 4/20 0.48
KMT2A Q03164 1/20 0.48
GAA P10253 2/20 0.47
HTT P42858 1/20 0.45
HPGD P15428 3/20 0.41
ALDH1A1 P00352 4/20 0.40
LMNA P02545 3/20 0.40
NPSR1 Q6W5P4 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GLA P06280 1/20 0.40
MAPK1 P28482 1/20 0.39
MAPK10 P53779 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10488534 0.91 SMN1; SMN2 (0.62) SMN1; SMN2PDE4DAURKAMAPTPOLB
SCHEMBL10488465 0.90 SMN1; SMN2 (0.61) SMN1; SMN2PDE4DAURKAMAPTPOLB
SCHEMBL10488587 0.89 SMN1; SMN2 (0.60) SMN1; SMN2PDE4DAURKAMAPTPOLB
SCHEMBL10488562 0.89 SMN1; SMN2 (0.60) SMN1; SMN2PDE4DAURKAMAPTPOLB
SCHEMBL10488962 0.88 SMN1; SMN2 (0.68) SMN1; SMN2PDE4DAURKAMAPTPOLB
SCHEMBL10488577 0.84 SMN1; SMN2 (0.57) SMN1; SMN2PDE4DAURKAMAPTPOLB
SCHEMBL10489006 0.83 PDE4D (0.67) SMN1; SMN2PDE4DAURKAMAPTPOLB
SCHEMBL10488470 0.83 SMN1; SMN2 (0.48) SMN1; SMN2PDE4DAURKAKDM4EGAA
Hydrochloric Acid SCHEMBL10488574 0.83 SMN1; SMN2 (0.56) SMN1; SMN2PDE4DAURKAMAPTPOLB
SCHEMBL10488922 0.82 SMN1; SMN2 (0.62) SMN1; SMN2PDE4DAURKAMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4826866-A 3-amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants, muscle relaxants and anxiolytics A. H. ROBINS COMPANY, INCORPORATED (US) 1989-05-02 US claimed
EP-0315433-A2 3-amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants, muscle relaxants and anxiolytics A.H. ROBINS COMPANY, INCORPORATED (US) 1989-05-10 EP disclosed