SCHEMBL10490758

SCHEMBL10490758

O=C(OCc1ccc([N+](=O)[O-])cc1)Oc1c[c]ccc1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.58
RAB9A P51151 3/20 0.46
AKR1C3 P42330 1/20 0.45
MAOB P27338 2/20 0.44
MAOA P21397 1/20 0.44
HTT P42858 2/20 0.43
MAPT P10636 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
IDO1 P14902 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10490876 0.84 HTR2A (0.67) HTR2ARAB9AAKR1C3MAOBHTT
SCHEMBL10490891 0.83 KMT2A (0.50) HTTMAPTNPSR1L3MBTL1
SCHEMBL5827968 0.82 HTR2A (0.80) HTR2ARAB9AAKR1C3MAOBHTT
SCHEMBL23042226 0.82 HTR2A (0.67) HTR2ARAB9AAKR1C3MAOBIDO1
SCHEMBL29074496 0.81 MAPT (0.58) RAB9AAKR1C3MAOBMAOAMAPT
SCHEMBL10490867 0.81 HTR2A (0.53) HTR2ARAB9AAKR1C3MAOBHTT
SCHEMBL5719541 0.80 HTT (0.56) RAB9AAKR1C3MAOBMAOAHTT
SCHEMBL14621621 0.79 HTR2A (0.74) HTR2ARAB9AAKR1C3MAOBHTT
SCHEMBL1714950 0.79 HTR2A (0.70) HTR2ARAB9AHTTMAPT
Water SCHEMBL10938437 0.78 HTR2A (0.73) HTR2ARAB9AMAOBHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0219926-A2 Cephalosporins, processes for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1987-04-29 EP claimed
US-4835150-A ANTIBIOTICS BEECHAM GROUP P.L.C. (GB) 1989-05-30 US disclosed
EP-0308559-A2 Cephalosporins, process for their preparation, pharmaceutical compositions containing them and intermediates BEECHAM GROUP PLC (GB) 1989-03-29 EP disclosed
EP-0265185-A2 Cephalosporins, processes for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1988-04-27 EP disclosed
EP-0219926-A2 Cephalosporins, processes for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1987-04-29 EP disclosed