SCHEMBL10495679

SCHEMBL10495679

NC(=O)c1c(Br)cc(Br)c(O)c1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA4 P22748 2/20 0.44
CA6 P23280 2/20 0.44
TTR P02766 1/20 0.40
GPR35 Q9HC97 2/20 0.38
PTPN1 P18031 3/20 0.37
TSHR P16473 2/20 0.37
CYP3A4 P08684 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MAP2K1 Q02750 1/20 0.36
AKR1C4 P17516 1/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
AKR1C1 Q04828 1/20 0.36
AKR1B1 P15121 1/20 0.35
ERN1 O75460 1/20 0.35
MAPT P10636 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30009277 0.80 TTR (0.52) CA1CA2CA4CA6TTR
SCHEMBL124390 0.80 TTR (0.52) CA1CA2CA4CA6TTR
SCHEMBL10495686 0.78 CA1 (0.37) CA1CA2CA4CA6TTR
SCHEMBL31320039 0.77 CA1 (0.43) CA1CA2CA4CA6TTR
SCHEMBL10964657 0.74 ERN1 (0.43) CA1CA2CA4CA6TTR
SCHEMBL69904 0.72 CA1 (0.67) CA1CA2CA4CA6TTR
SCHEMBL1003689 0.72 TSHR (0.43) CA1CA2GPR35TSHRCYP3A4
SCHEMBL10495740 0.71 CSNK2A2 (0.34) MAP2K1AKR1B1
SCHEMBL28017537 0.70 CA1 (0.63) CA1CA2CA4CA6TTR
SCHEMBL4351080 0.70 TTR (0.62) TTRTSHRCYP3A4TDP1MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4869913-A DIETETICS SCHERING AKTIENGESELLSCHAFT (DE) 1989-09-26 US disclosed
US-4522839-A 3-Substituted 2,4,6-trihalogenated benzamides as sweetening agents SCHERING AKTIENGESELLSCHAFT (DE) 1985-06-11 US disclosed
EP-0055689-B1 3-SUBSTITUTED 2,4,6-TRIHALOGENOBENZAMIDES AND THEIR SALTS, THEIR PREPARATION AND THEIR USE AS SUBSTITUTES FOR NATURAL SWEETENING AGENTS, AND SWEETENERS CONTAINING THEM SCHERING AKTIENGESELLSCHAFT (DE) 1984-07-04 EP disclosed
US-4429152-A DIABETES, DIETETICS SCHERING, AKTIENGESELLSCHAFT (DE) 1984-01-31 US disclosed
EP-0055689-A1 3-Substituted 2,4,6-trihalogenobenzamides and their salts, their preparation and their use as substitutes for natural sweetening agents, and sweeteners containing them SCHERING AKTIENGESELLSCHAFT (DE) 1982-07-07 EP disclosed