SCHEMBL10964657

SCHEMBL10964657

NC(=O)c1cc(Br)c(O)c(Br)c1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.43
KDM4E B2RXH2 3/20 0.42
MAPT P10636 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
AKR1C4 P17516 2/20 0.41
AKR1C3 P42330 2/20 0.41
AKR1C2 P52895 2/20 0.41
AKR1C1 Q04828 2/20 0.41
TTR P02766 1/20 0.40
AKR1B1 P15121 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
DGAT1 O75907 1/20 0.38
GPR35 Q9HC97 2/20 0.38
PTPN1 P18031 3/20 0.37
TSHR P16473 2/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7950797 0.87 AKR1B1 (0.43) ERN1KDM4EMAPTMEN1KMT2A
SCHEMBL29593387 0.80 AKR1C3 (0.63) KDM4EAKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL4891804 0.80 AKR1C3 (0.63) KDM4EAKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL895511 0.78 AKR1C4 (0.67) ERN1KDM4EMAPTMEN1KMT2A
SCHEMBL4072963 0.78 ALDH1A1 (0.43) KDM4EMAPTMEN1KMT2AAKR1C4
SCHEMBL16644420 0.76 DGAT1 (0.46) ERN1KDM4EMAPTMEN1KMT2A
SCHEMBL3238108 0.75 GSK3B (0.41) KDM4EMAPTMEN1KMT2AAKR1C4
SCHEMBL10495679 0.74 CA1 (0.44) ERN1MAPTMEN1KMT2AAKR1C4
SCHEMBL31700545 0.74 ERN1 (0.61) ERN1KDM4EMAPTMEN1KMT2A
SCHEMBL19423432 0.74 HSD17B10 (0.47) ERN1KDM4EMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0075881-B1 7-DEAZAPURINE DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 1985-02-13 EP disclosed
US-4435570-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1984-03-06 US disclosed
EP-0075881-A1 7-Deazapurine derivatives Takeda Chemical Industries, Ltd. (JP) 1983-04-06 EP disclosed