SCHEMBL10500802

SCHEMBL10500802

C1=CC(c2ccco2)C=CN1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 10/20 0.40
CHRM3 P20309 10/20 0.40
CHRM1 P11229 9/20 0.40
CHRM2 P08172 9/20 0.40
CHRM4 P08173 9/20 0.40
ALDH1A1 P00352 5/20 0.39
KMT2A Q03164 4/20 0.39
POLB P06746 3/20 0.39
MAPT P10636 3/20 0.39
MEN1 O00255 3/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 2/20 0.39
BLM P54132 2/20 0.39
USP2 O75604 1/20 0.39
THRB P10828 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
NR4A1 P22736 1/20 0.39
MAPK1 P28482 1/20 0.39
BRCA1 P38398 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23316883 0.65 ALDH1A1 (0.47) CHRM5CHRM3CHRM1CHRM2CHRM4
SCHEMBL8462330 0.65
SCHEMBL18966709 0.64 CHRM5 (0.57) CHRM5CHRM3CHRM1CHRM2CHRM4
SCHEMBL503332 0.62 RECQL (0.34) ALDH1A1HPGDHSD17B10ALOX12TDP1
SCHEMBL21402172 0.62
SCHEMBL9534606 0.61 ALDH1A1 (0.46) CHRM5CHRM3CHRM1CHRM2CHRM4
SCHEMBL5334097 0.61 CHRM5 (0.44) CHRM5CHRM3CHRM1CHRM2CHRM4
SCHEMBL30987970 0.61 ALDH1A1 (0.55) CHRM5CHRM3CHRM1CHRM2CHRM4
SCHEMBL10491245 0.61 CHRM5 (0.44) CHRM5CHRM3CHRM1CHRM2CHRM4
SCHEMBL7386543 0.61 RECQL (0.33) ALDH1A1HPGDHSD17B10ALOX12TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0088903-B1 1,4-DIHYDROPYRIDINE-3,5-DICARBOXYLIC ACID ESTER DERIVATIVES Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1988-11-23 EP claimed
US-4841054-A A LOW TOXICITY, HIGH STABILITY MEDICATION FOR HYPERTENSIVE ACTIVITY INSTITUTE ORGANICHESKOGO SINTEZA AKADEMII NAUK LATVISISKOI SSR 1989-06-20 US disclosed