SCHEMBL1050281

SCHEMBL1050281

O=Cc1cccc(OCc2ccccc2)c1OCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 1/20 0.59
CDK1 P06493 1/20 0.59
CDK4 P11802 1/20 0.59
CCNB1 P14635 1/20 0.59
CCND1 P24385 1/20 0.59
CCNB3 Q8WWL7 1/20 0.59
L3MBTL1 Q9Y468 3/20 0.51
MAPT P10636 2/20 0.51
TDP1 Q9NUW8 2/20 0.51
MAPK1 P28482 1/20 0.51
SMN1; SMN2 Q16637 2/20 0.50
PTGER1 P34995 2/20 0.50
PTGER4 P35408 2/20 0.50
PTGER3 P43115 2/20 0.50
PTGER2 P43116 2/20 0.50
ALDH1A1 P00352 1/20 0.50
HPGD P15428 1/20 0.50
HTT P42858 1/20 0.50
SRC P12931 1/20 0.49
NPC1 O15118 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL411835 0.91 HTR1A (0.56) CCNB2CDK1CDK4CCNB1CCND1
Perchlorate SCHEMBL10994108 0.90 CCNB2 (0.50) CCNB2CDK1CDK4CCNB1CCND1
SCHEMBL28877513 0.90 CCNB2 (0.53) CCNB2CDK1CDK4CCNB1CCND1
SCHEMBL28788684 0.90 CCNB2 (0.52) CCNB2CDK1CDK4CCNB1CCND1
SCHEMBL4294807 0.89 CCNB2 (0.55) CCNB2CDK1CDK4CCNB1CCND1
SCHEMBL1125006 0.89 KDM4E (0.60) CCNB2CDK1CDK4CCNB1CCND1
SCHEMBL28129638 0.89 KDM4E (0.60) CCNB2CDK1CDK4CCNB1CCND1
SCHEMBL16632680 0.88 KMT2A (0.54) CCNB2CDK1CDK4CCNB1CCND1
SCHEMBL5839420 0.87 CCNB2 (0.51) CCNB2CDK1CDK4CCNB1CCND1
SCHEMBL433401 0.86 CCNB2 (0.72) CCNB2CDK1CDK4CCNB1CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 136 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4663636-A2 TRIFLUOROMETHYL SUBSTITUTED PYRAZOLES AS HUMAN PLASMA KALLIKREIN INHIBITORS BioCryst Pharmaceuticals, Inc. (US) 2025-12-17 EP disclosed
US-20250270171-A1 HUMAN PLASMA KALLIKREIN INHIBITORS WILMINGTON TRUST, NATIONAL ASSOCIATION 2025-08-28 US disclosed
US-20250257040-A1 HUMAN PLASMA KALLIKREIN INHIBITORS WILMINGTON TRUST, NATIONAL ASSOCIATION 2025-08-14 US disclosed
EP-4180424-B1 SUBSTITUTED PYRAZOLES AS HUMAN PLASMA KALLIKREIN INHIBITORS BIOCRYST PHARM INC (US) 2025-06-25 EP disclosed
US-12162838-B2 Human plasma kallikrein inhibitors BIOCRYST PHARMACEUTICALS, INC. (US) 2024-12-10 US disclosed
US-12116346-B2 Human plasma kallikrein inhibitors BIOCRYST PHARMACEUTICALS, INC. (US) 2024-10-15 US disclosed
EP-3274322-B1 STABLE COMPOSITIONS FOR PREVENTION / PROPHYLACTIC TREATMENT OF POISON IVY DERMATITIS THE UNIV OF MISSISSIPPI (US) 2024-08-14 EP disclosed
CN-113307772-B Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2024-06-28 CN disclosed
US-20240150296-A1 HUMAN PLASMA KALLIKREIN INHIBITORS WILMINGTON TRUST, NATIONAL ASSOCIATION 2024-05-09 US disclosed
US-20240150295-A1 HUMAN PLASMA KALLIKREIN INHIBITORS WILMINGTON TRUST, NATIONAL ASSOCIATION 2024-05-09 US disclosed
WO-1995013262-A1 SUBSTITUTED PHENYL COMPOUNDS RHONE-POULENC RORER LIMITED (GB) 1995-05-18 WO disclosed
EP-0228625-B1 PEPTIDE DERIVATIVES INHIBITORS OF HYDROXYLING ENZYMES, THEIR PROCESS OF PREPARATION, THE AGENTS THEREOF AND THEIR USE HOECHST AKTIENGESELLSCHAFT (DE) 1992-01-02 EP disclosed
EP-0401517-A1 Substituted 2-alkynylphenols with anti-inflammatory action, a process for their preparation and pharmaceutical compositions thereof CAMILLO CORVI S.p.A. (IT) 1990-12-12 EP disclosed
EP-0339927-A2 Amide compounds their production and use Takeda Chemical Industries, Ltd. (JP) 1989-11-02 EP disclosed
US-4797471-A INHIBITING COLAGEN SYNTHESIS HOECHST AKTIENGESELLSCHAFT (DE) 1989-01-10 US disclosed
EP-0228625-A2 Peptide derivatives inhibitors of hydroxyling enzymes, their process of preparation, the agents thereof and their use HOECHST AKTIENGESELLSCHAFT (DE) 1987-07-15 EP disclosed
EP-0189142-A2 Arylalkoxyphenyl-allylic alcohols as agents for the treatment of hypersensitive ailments USV PHARMACEUTICAL CORPORATION (US) 1986-07-30 EP disclosed
US-4529811-A Process for isolating organic compounds and lithium salt complexes useful in said process G. D. SEARLE & CO. (US) 1985-07-16 US disclosed
US-4054617-A LEATHER PROCESSING DIAMOND SHAMROCK CORPORATION (US) 1977-10-18 US disclosed
US-3934975-A Leather treating process DIAMOND SHAMROCK CORPORATION (US) 1976-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12116346-B2 Human plasma kallikrein inhibitors KLKB1, KLK5, KLK1 CCNB2 3540/4885CDK1 1651/4885CDK4 4605/4885
US-20250270171-A1 HUMAN PLASMA KALLIKREIN INHIBITORS KLKB1, KLK5, KLK1 CCNB2 3540/4885CDK1 1651/4885CDK4 4605/4885
US-20240150296-A1 HUMAN PLASMA KALLIKREIN INHIBITORS KLKB1, KLK5, KLK1 CCNB2 3540/4885CDK1 1651/4885CDK4 4605/4885
US-20240150295-A1 HUMAN PLASMA KALLIKREIN INHIBITORS KLKB1, KLK5, KLK1 CCNB2 3540/4885CDK1 1651/4885CDK4 4605/4885
US-20250257040-A1 HUMAN PLASMA KALLIKREIN INHIBITORS KLKB1, KLK5, KLK1 CCNB2 3540/4885CDK1 1651/4885CDK4 4605/4885
US-12162838-B2 Human plasma kallikrein inhibitors KLKB1, KLK5, KLK1 CCNB2 3540/4885CDK1 1651/4885CDK4 4605/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.