SCHEMBL10502811

SCHEMBL10502811

O=C(O)CCc1cccc2c1Sc1cc(C(=O)O)ccc1CC2

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 2/20 0.39
SRD5A1 P18405 1/20 0.39
LTB4R Q15722 1/20 0.37
PTGER4 P35408 10/20 0.36
PTGER2 P43116 10/20 0.36
PTGER1 P34995 1/20 0.36
PTGER3 P43115 1/20 0.36
ALDH1A1 P00352 1/20 0.36
APEX1 P27695 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10503522 0.75 RXRB (0.38) SRD5A2SRD5A1ALDH1A1APEX1RXRA
SCHEMBL9681571 0.74 SRD5A2 (0.54) SRD5A2SRD5A1ALDH1A1RXRA
SCHEMBL27794501 0.68 SRD5A2 (0.58) SRD5A2SRD5A1ALDH1A1RXRA
SCHEMBL10502889 0.66 ALDH1A1 (0.62) SRD5A2SRD5A1ALDH1A1RXRARXRB
SCHEMBL11098487 0.65 ALDH1A1 (0.41) SRD5A2SRD5A1ALDH1A1RXRARXRB
SCHEMBL27151108 0.65 ALDH1A1 (0.46) SRD5A2SRD5A1ALDH1A1
SCHEMBL7825857 0.65 MEN1 (0.49) ALDH1A1RXRARXRBRXRG
SCHEMBL10784805 0.64 NPSR1 (0.47) LTB4RPTGER4PTGER2PTGER1PTGER3
SCHEMBL9778275 0.64 MAPT (0.46) SRD5A2SRD5A1ALDH1A1
SCHEMBL11015563 0.64 ALDH1A1 (0.42) SRD5A2SRD5A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0138533-B1 6H-DIBENZ(B,F)THIEPIN COMPOUNDS MERCK FROSST CANADA INC. (CA) 1989-04-12 EP disclosed
US-4622403-A ALLERGIC CONDITIONS MERCK FROSST CANADA, INC. (CA) 1986-11-11 US disclosed
EP-0138533-A2 6H-dibenz(b,f)thiepin compounds MERCK FROSST CANADA INC. (CA) 1985-04-24 EP disclosed