SCHEMBL10508186

SCHEMBL10508186

NC(=O)Cc1cc(-c2ccccc2)nc2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.58
LMNA P02545 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
PDE10A Q9Y233 1/20 0.58
ACACA Q13085 3/20 0.56
DHODH Q02127 1/20 0.55
ACHE P22303 1/20 0.54
CYP2C9 P11712 1/20 0.54
TACR3 P29371 3/20 0.51
CYP3A4 P08684 1/20 0.50
HPGD P15428 2/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
POLB P06746 2/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
NPC1 O15118 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10506477 0.87 KDM4E (0.61) KDM4ELMNASMN1; SMN2PDE10AACACA
SCHEMBL10509237 0.85 KDM4E (0.55) KDM4ELMNASMN1; SMN2PDE10AACACA
SCHEMBL13268004 0.81 KDM4E (0.54) KDM4ELMNASMN1; SMN2PDE10ADHODH
SCHEMBL1259674 0.80 ACHE (0.59) KDM4ELMNASMN1; SMN2PDE10AACACA
SCHEMBL13821792 0.79 PLA2G10 (0.48) KDM4ESMN1; SMN2ACACAACHECYP3A4
SCHEMBL2998020 0.79 KDM4E (0.50) KDM4EACACAACHECYP3A4HPGD
SCHEMBL10675180 0.79 KDM4E (0.76) KDM4ELMNASMN1; SMN2PDE10ACYP2C9
SCHEMBL10677865 0.79 KDM4E (0.54) KDM4ELMNASMN1; SMN2PDE10ADHODH
SCHEMBL13243228 0.78 ESRRB (0.59) KDM4ELMNASMN1; SMN2PDE10AACACA
SCHEMBL3968020 0.78 ACHE (0.58) KDM4ELMNASMN1; SMN2PDE10AACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0210084-B1 AMIDES, PROCESSES FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM RHONE-POULENC SANTE (FR) 1989-02-08 EP disclosed
EP-0210084-A1 Amides, processes for their preparation and medicaments containing them RHONE-POULENC SANTE (FR) 1987-01-28 EP disclosed