SCHEMBL10508576

SCHEMBL10508576

NS(=O)(=O)c1cc2cc(O)c(O)cc2o1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 16/20 0.66
CA12 O43570 2/20 0.46
CA9 Q16790 2/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
CYP1A2 P05177 1/20 0.46
BCHE P06276 1/20 0.46
GLA P06280 1/20 0.46
CYP3A4 P08684 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
AKR1B1 P15121 1/20 0.46
HPGD P15428 1/20 0.46
ALOX15 P16050 1/20 0.46
ACHE P22303 1/20 0.46
PTGS1 P23219 1/20 0.46
CASP1 P29466 1/20 0.46
XDH P47989 1/20 0.46
CASP7 P55210 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10509194 0.83 CA2 (0.59) CA2CA12CA9KDM4EALDH1A1
SCHEMBL10509670 0.81 CA2 (0.57) CA2CA12CA9KDM4EALDH1A1
SCHEMBL10508948 0.79 CA2 (1.00) CA2CA12CA9KDM4EALDH1A1
SCHEMBL10509061 0.79 CA2 (1.00) CA2CA12CA9KDM4EALDH1A1
SCHEMBL10510393 0.76 CA2 (0.64) CA2CA12CA9KDM4EALDH1A1
SCHEMBL10508066 0.74 CA2 (0.51) CA2CA12CA9PTGS1
SCHEMBL9424948 0.73 PIM1 (0.55) CA12CA9KDM4EALDH1A1LMNA
SCHEMBL1156380 0.72 CA2 (1.00) CA2CA12CA9KDM4EAKR1B1
SCHEMBL29926951 0.72 CA2 (1.00) CA2CA12CA9KDM4EAKR1B1
SCHEMBL10993963 0.72 CA2 (0.64) CA2CA12CA9LMNACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0152340-B1 2-Sulfamoylbenzo[b]furan derivatives and ophtalmic composition for the treatment of elevated intraocular pressure MERCK & CO. INC. (US) 1989-05-10 EP disclosed
US-4544667-A CARBONIC ANHYDRASE INHIBITOR; VISION DEFECTS MERCK & CO., INC. (US) 1985-10-01 US disclosed
EP-0152340-A1 2-Sulfamoylbenzo[b]furan derivatives and ophtalmic composition for the treatment of elevated intraocular pressure MERCK & CO. INC. (US) 1985-08-21 EP disclosed