SCHEMBL10517455

SCHEMBL10517455

COc1ccc(-c2[nH]c(=O)c(C(=O)O)cc2-c2ccc(OCc3ccccc3)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSTP1 P09211 2/20 0.51
MAPT P10636 1/20 0.50
MAPK1 P28482 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
NOD2 Q9HC29 1/20 0.50
MCL1 Q07820 1/20 0.50
SMN1; SMN2 Q16637 4/20 0.49
RXFP1 Q9HBX9 2/20 0.49
RAB9A P51151 2/20 0.49
TP53 P04637 1/20 0.49
PKM P14618 1/20 0.49
NFKB1 P19838 1/20 0.49
NFKB2 Q00653 1/20 0.49
RELA Q04206 1/20 0.49
MRGPRX4 Q96LA9 1/20 0.49
DHODH Q02127 3/20 0.48
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
NPC1 O15118 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5904153 0.87 KDM4E (0.59) SMN1; SMN2RXFP1KDM4EALDH1A1GAA
SCHEMBL10517403 0.86 KCNH2 (0.52) GSTP1MAPTNPSR1MCL1SMN1; SMN2
SCHEMBL10516469 0.85 KDM4E (0.54) MAPTSMN1; SMN2RXFP1TP53KDM4E
SCHEMBL10514341 0.82 GSK3B (0.54) MAPTSMN1; SMN2RXFP1KDM4EALDH1A1
SCHEMBL10483018 0.80 KDM4E (0.51) MAPTSMN1; SMN2RXFP1RAB9ATP53
SCHEMBL14867324 0.76 SERPINE1 (0.55) GSTP1MAPTMAPK1NPSR1NOD2
SCHEMBL14741167 0.75 KDM4E (0.57) MAPTSMN1; SMN2RXFP1KDM4EALDH1A1
SCHEMBL10515809 0.74 MAOB (0.48) MAPTNOD2MAOB
SCHEMBL7991836 0.73 DHODH (0.58) MAPTSMN1; SMN2RAB9ATP53DHODH
SCHEMBL6799282 0.73 MCL1 (0.63) GSTP1MCL1DHODHFFAR1FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308020-A2 5-(aryl and heteroaryl)-6-(aryl and heteroaryl)-1,2-dihydro-2-oxo 3-pyridinecarboxylic acids and derivatives thereof MERCK & CO. INC. (US) 1989-03-22 EP claimed