SCHEMBL10519065

SCHEMBL10519065

CC1CC(=O)NN=C1c1ccc2oc(N3CCNCC3)nc2c1

nearest known ligand 0.85

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 16/20 0.85
PDE3B Q13370 3/20 0.50
PDE3A Q14432 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2583140 0.92 GPR119 (1.00) GPR119
SCHEMBL10522354 0.92 GPR119 (0.83) GPR119PDE3BPDE3A
SCHEMBL10520468 0.90 GPR119 (0.70) GPR119PDE3BPDE3A
SCHEMBL10519406 0.85 GPR119 (0.64) GPR119
SCHEMBL2590468 0.83 GPR119 (0.98) GPR119
SCHEMBL2590391 0.82 GPR119 (1.00) GPR119
SCHEMBL2590176 0.82 GPR119 (0.83) GPR119PDE3BPDE3A
SCHEMBL2590196 0.82 GPR119 (1.00) GPR119PDE3BPDE3A
SCHEMBL2584523 0.81 GPR119 (1.00) GPR119
SCHEMBL7331168 0.80 GPR119 (0.62) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0196005-B1 PYRIDAZINONES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1989-12-20 EP disclosed
EP-0196005-A1 Pyridazinones, their preparation and pharmaceutical compositions containing them Dr. Karl Thomae GmbH (DE) 1986-10-01 EP disclosed