SCHEMBL10522160

SCHEMBL10522160

CCN1CCCCC1CCN(C)CC(=O)N1c2ccccc2C(=O)Nc2cccnc21

nearest known ligand 0.75

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.68
CYP3A4 P08684 1/20 0.68
CHRM2 P08172 1/20 0.68
CHRM4 P08173 1/20 0.68
CHRM1 P11229 1/20 0.68
CHRM3 P20309 1/20 0.68
MAPK1 P28482 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10459903 0.91 CHRM2 (0.62) CYP1A2CYP3A4CHRM2CHRM4CHRM1
SCHEMBL8879186 0.91 CHRM2 (0.61) CYP1A2CYP3A4CHRM2CHRM4CHRM1
SCHEMBL9803290 0.90 CYP1A2 (0.69) CYP1A2CYP3A4CHRM2CHRM4CHRM1
SCHEMBL10514973 0.90 CYP1A2 (0.55) CYP1A2CYP3A4CHRM2CHRM4CHRM1
Hydrochloric Acid SCHEMBL9803350 0.90 CYP1A2 (0.69) CYP1A2CYP3A4CHRM2CHRM4CHRM1
SCHEMBL8879790 0.89 CHRM2 (0.61) CYP1A2CHRM2CHRM4CHRM1CHRM3
Hydrochloric Acid SCHEMBL9870848 0.88 CHRM2 (0.60) CYP1A2CHRM2CHRM4CHRM1CHRM3
SCHEMBL10508829 0.87 CHRM2 (0.77) CYP1A2CYP3A4CHRM2CHRM4CHRM1
SCHEMBL10519813 0.87 CHRM2 (0.61) CYP1A2CYP3A4CHRM2CHRM4CHRM1
SCHEMBL10510299 0.86 CYP1A2 (0.85) CYP1A2CYP3A4CHRM2CHRM4CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0346744-A1 Condensed diazepinones, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1989-12-20 EP disclosed