SCHEMBL10537855

SCHEMBL10537855

COc1ccc(F)cc1NC(=O)NC1CC2CCC(C1)N2C

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.51
MEN1 O00255 2/20 0.51
ALDH1A1 P00352 2/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 2/20 0.48
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
POLB P06746 1/20 0.48
HTT P42858 1/20 0.47
HTR4 Q13639 1/20 0.47
DRD2 P14416 2/20 0.47
ADRA1D P25100 2/20 0.47
ADRA1A P35348 2/20 0.47
ADRA1B P35368 2/20 0.47
HTR3A P46098 2/20 0.46
USP2 O75604 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10540683 0.92 MAPT (0.55) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL10539603 0.88 MRGPRX1 (0.48) DRD2ADRA1DADRA1AADRA1BHTR3A
SCHEMBL10539974 0.87 MAPT (0.56) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL10540979 0.87 TSHR (0.59) KMT2AMEN1ALDH1A1GAAMAPT
Hydrochloric Acid SCHEMBL10538812 0.86 KMT2A (0.51) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL10755457 0.86 KMT2A (0.69) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL10542205 0.86 POLB (0.60) KMT2AALDH1A1MAPTKDM4ELMNA
SCHEMBL10541801 0.85 KMT2A (0.50) KMT2AMEN1ALDH1A1GAAMAPT
Hydrochloric Acid SCHEMBL10542169 0.85 KMT2A (0.68) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL10541780 0.85 CYP2D6 (0.54) KMT2AMEN1ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0235878-A2 Novel compounds BEECHAM GROUP PLC (GB) 1987-09-09 EP claimed
US-4797387-A ANALGESICS, ANTIEMETICS BEECHAM GROUP, P.L.C. (GB) 1989-01-10 US disclosed
EP-0235878-A2 Novel compounds BEECHAM GROUP PLC (GB) 1987-09-09 EP disclosed