SCHEMBL10543714

SCHEMBL10543714

CC(C)=CCCCCBr.[MgH2]

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.39
ALOX15 P16050 3/20 0.36
MEN1 O00255 2/20 0.36
CYP3A4 P08684 2/20 0.36
SQLE Q14534 3/20 0.35
MAPT P10636 2/20 0.34
ALDH1A1 P00352 2/20 0.34
TSHR P16473 1/20 0.34
UGT1A1 P22309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10542200 0.97
SCHEMBL10596935 0.95 KMT2A (0.39) KMT2AALOX15MEN1CYP3A4SQLE
SCHEMBL5883430 0.95 KMT2A (0.39) KMT2AALOX15MEN1CYP3A4SQLE
SCHEMBL4574808 0.89
SCHEMBL8078444 0.83 KMT2A (0.50) KMT2AALOX15MEN1CYP3A4SQLE
SCHEMBL7679632 0.80
SCHEMBL230243 0.77
SCHEMBL9633770 0.77 KMT2A (0.67) KMT2AALOX15MEN1CYP3A4SQLE
SCHEMBL11131196 0.76 KMT2A (0.50) KMT2AALOX15MEN1CYP3A4SQLE
SCHEMBL31399494 0.74 DGKA (0.44) ALOX15CYP3A4ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4822804-A 5,6,7,-trinor-4,8-inter-m-phenylene 2-nor PGI2 derivatives and anti-ulcer, anti-thrombotic and anti-hypertensive pharmaceutical compositions containing them TORAY INDUSTRIES, INC. (JP) 1989-04-18 US disclosed
EP-0060640-B1 5,6,7-TRINOR-4,8-INTER-M-PHENYLENE PGI DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM TORAY INDUSTRIES, INC. (JP) 1985-11-13 EP disclosed
EP-0060640-A1 5,6,7-Trinor-4,8-inter-m-phenylene PGI derivatives and pharmaceutical compositions containing them TORAY INDUSTRIES, INC. (JP) 1982-09-22 EP disclosed