SCHEMBL10546321

SCHEMBL10546321

N#CCCc1cc(F)cc(F)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
IDO1 P14902 2/20 0.38
DAO P14920 2/20 0.37
MPO P05164 1/20 0.34
SLC6A4 P31645 1/20 0.34
CYP17A1 P05093 1/20 0.32
CYP21A2 P08686 1/20 0.32
CYP11B1 P15538 1/20 0.32
THRB P10828 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA9 Q16790 1/20 0.31
TAAR1 Q96RJ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22165081 0.86 MEN1 (0.44) MEN1KMT2AIDO1MPOSLC6A4
SCHEMBL24289637 0.86 MEN1 (0.44) MEN1KMT2AMPOSLC6A4
SCHEMBL25709303 0.81 MEN1 (0.40) MEN1KMT2AMPOSLC6A4
SCHEMBL28049281 0.80 MEN1 (0.47) MEN1KMT2AMPOSLC6A4
SCHEMBL31210245 0.79 MEN1 (0.50) MEN1KMT2AMPOSLC6A4THRB
SCHEMBL2023893 0.79 MEN1 (0.73) MEN1KMT2AIDO1DAOSLC6A4
SCHEMBL5546168 0.76 DAO (0.40) IDO1DAOCYP17A1CYP21A2CYP11B1
SCHEMBL21728102 0.76 IDO1 (0.38) IDO1DAOCYP17A1CYP21A2CYP11B1
SCHEMBL4847285 0.76 DAO (0.40) IDO1DAOCYP17A1CYP21A2CYP11B1
SCHEMBL2023212 0.76 MEN1 (0.52) MEN1KMT2AIDO1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4859779-A ENZYME INHIBITORS SMITHKLINE BECKMAN CORPORATION (US) 1989-08-22 US disclosed
US-4837353-A 2-/N-PHENYLALKYL-N-FORMYL/AMINO-3-HYDROXY-2-PROPENOIC ACID DERIVATIVES SMITHKLINE BECKMAN CORPORATION (US) 1989-06-06 US disclosed
EP-0284375-A1 Dopamine-beta-hydroxylase inhibitors SMITHKLINE BEECHAM CORPORATION (US) 1988-09-28 EP disclosed
US-4762850-A Dopamine-beta-hydroxylase inhibitors SMITHKLINE BECKMAN CORPORATION (US) 1988-08-09 US disclosed